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3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(methylsulfanyl)phenyl]urea
3-(2,5-dimethoxyphenyl)-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidine
N-[(1-propylpyrrolidin-3-yl)methyl]-3-azaspiro[5.5]undecan-9-amine
5-{8-benzyl-2,8-diazaspiro[5.5]undecan-2-yl}-1-(3-methylbutyl)azepan-2-one
2-chloro-N-[2-(1,2,3-thiadiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
N,3-dimethyl-N-[2-(oxan-2-yl)ethyl]-5-propyl-1-benzofuran-2-carboxamide
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
5-(phenoxymethyl)-N-[(4-phenyloxan-4-yl)methyl]-1H-pyrazole-3-carboxamide
N,3,5-trimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-{4-[4-(2-ethylpiperidine-1-carbonyl)phenoxy]piperidin-1-yl}-2-methoxyethan-1-one
2-{4-[({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]piperidin-1-yl}ethan-1-ol
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-N-(3-fluorophenyl)piperidin-3-amine
4-[(1-{[3-(furan-2-yl)phenyl]methyl}piperidin-2-yl)methyl]morpholine
4-fluoro-N-{2-[(4-hydroxy-2-phenylpyrimidin-5-yl)formamido]ethyl}benzamide
1-(2,1,3-benzoxadiazol-5-ylmethyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
(2S)-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
dimethyl[3-(2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenoxy)propyl]amine
1-(1H-indazol-6-yl)-4-[3-(pyridin-3-yl)propanoyl]piperazin-2-one
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-ethyl-1,3,4-thiadiazol-2-yl)piperidine
2-(2H-1,2,3-benzotriazol-2-yl)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N-methylbenzamide
2-(8-{[2-(furan-2-yl)phenyl]methyl}-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl)acetamide
(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-(thiophen-2-yl)-1H-pyrazol-4-yl)methanol
N-[3-(3-methoxyphenyl)phenyl]-1-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
3-{[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amino}propane-1,2-diol
2-({6-[(cyclopent-3-en-1-yl)amino]pyrazin-2-yl}sulfanyl)acetic acid
methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
N-[(1R,3R)-3-aminocyclopentyl]-6-(4-methoxyphenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
2-(3-methyl-1,2-oxazol-5-yl)-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}acetamide
2-(2,1,3-benzothiadiazol-5-ylmethyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
9-(pyrrolidine-1-sulfonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
5-({4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
4-(1H-pyrazol-1-yl)-1-(thiophene-3-carbonyl)piperidine-4-carboxylic acid
N-cyclopropyl-1-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carboxamide
3-methanesulfonamido-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
4-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]-N,N-dimethylpiperazine-1-carboxamide
N-[(2S)-4-methyl-1-oxo-1-[4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pentan-2-yl]acetamide
2-(oxolan-2-ylmethyl)-4-[4-(thiophen-2-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-5-ethyl-N,2-dimethylpyrimidin-4-amine
N-(cyclohex-1-en-1-ylmethyl)-6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-(2,4-difluorophenyl)-1-[1-(pyridin-2-ylmethyl)azepan-3-yl]urea
6-(aminomethyl)-2-methyl-N-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]pyrimidin-4-amine
1-(4-methylphenyl)-4-[2-(methylsulfanyl)benzoyl]piperazin-2-one
1-[(2-chloro-6-fluoro-3-methoxyphenyl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-hydroxy-2-(pyridin-4-yl)ethyl]benzamide
(3S,4S)-1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol