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(2S,4S)-4-(2,6-difluoro-4-methoxybenzamido)-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
(1S,5R)-3-[4-(propan-2-yl)pyrimidin-2-yl]-3,9-diazabicyclo[3.3.2]decan-10-one
(3R,5S)-N-[(2,4-difluorophenyl)methyl]-1-(pyridin-3-ylmethyl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
(1S,5R)-6-benzyl-3-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-N'-(2-methylphenyl)propanediamide
5-methyl-N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]-1,2-oxazole-3-carboxamide
N-(furan-3-ylmethyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
1-{3-[2-(3-phenyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-4-phenylbenzamide
2-amino-6-cyclopropyl-4-(6-methoxy-1H-indazol-3-yl)pyridine-3-carbonitrile
3-(methoxymethyl)-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
ethyl 5-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
1-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}-4-(propan-2-yl)piperazine
3-{[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)sulfamoyl}-N-(pyridin-3-yl)benzamide
3-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-3,3,3-trifluoropropan-1-one
1-(4-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N5-[(2-benzyl-1,3-thiazol-4-yl)methyl]-N6-cyclopropyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
6-ethyl-2-(3-{[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
(2,3-dihydro-1-benzofuran-5-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methylpyridine-3-carboxylic acid
3-[2-(2,6-difluorophenyl)ethyl]-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
8-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
2-[5-(isoquinolin-5-yl)-4-phenyl-1H-imidazol-1-yl]-N-methylbutanamide
2-{1-cyclopentyl-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
2-methyl-4-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}butan-2-ol
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
2-(ethylamino)-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4-methyl-1,3-thiazole-5-carboxamide
4-[(6-methylpyridin-3-yl)oxy]-1-(6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidine-4-carboxylic acid
2-{6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}-1H-1,3-benzodiazole
N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)propanamide
methyl[1-(1,2-oxazol-3-yl)ethyl]{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
3-methyl-8-[1-(4-methylphenyl)cyclopropanecarbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(2-methylpropyl)amine
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-[(4-hydroxypiperidin-1-yl)methyl]piperidin-2-one
8-fluoro-2-{[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}quinolin-4-ol
2-[4-(1H-pyrazol-1-yl)phenyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetic acid
N-[(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]acetamide
N-[2-(2-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoacetyl)phenyl]propanamide
N'-(3,5-dimethylphenyl)-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)propanediamide
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-[2-(4-methoxyphenyl)ethyl]-1-methyl-N-(pyridin-3-ylmethyl)azepane-2-carboxamide
3-{[2-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl](methyl)amino}-1λ6-thiolane-1,1-dione
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
3,3-diphenyl-1-[(2S)-pyrrolidine-2-carbonyl]piperidine
1-methyl-N-(2-phenylpropan-2-yl)-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-cyclopropyl-1-(2-{1-[2-(2-methoxyphenyl)acetyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide