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[(3R,4R)-4-(azepan-1-ylmethyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methanol
(3R,4R)-3-cyclopropyl-1-[3-(4-fluorophenyl)benzoyl]-4-methylpyrrolidin-3-ol
4-[3-(methylsulfanyl)propyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[5-(3-cyclohexyl-1H-pyrazol-4-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
9-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-6-oxa-9-azaspiro[4.5]decane
3-(1-methyl-1H-pyrrol-2-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-5-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
4-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-5-methyl-1-propyl-1H-pyrazole
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N,5-dimethylimidazo[1,2-a]pyridine-2-carboxamide
1-[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
4-[1-(3-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]butanamide
1-[1-ethyl-3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-phenoxypropan-1-one
3-({1-[2-(3-chloro-4-hydroxyphenyl)acetyl]pyrrolidin-3-yl}methyl)benzamide
N,N-dimethyl-5-{[4-(3-phenylpropyl)-1,4-diazepan-1-yl]methyl}pyrimidin-2-amine
2-amino-6-{4-[(dimethylamino)methyl]thiophen-2-yl}-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
2-{2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
7-(3-phenylpropyl)-2-[2-(pyridin-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-methyl-4-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]piperazine-2-carboxylic acid
3-{[2-(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
N-[(5-fluoro-2-methylphenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-[2-(pyridin-2-ylmethoxy)phenyl]urea
(4-{[1-(1,3-benzothiazole-6-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
3-(3-aminopropyl)-7-fluoro-3,4-dihydroquinazolin-4-one
3,5-dimethyl-N-(oxan-4-ylmethyl)-1-benzofuran-2-carboxamide
1-(1-{2-[methyl(propan-2-yl)amino]acetyl}piperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide
2-cyclopentyl-8-[(1-propyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1λ6-thiane-1,1-dione
2-[(4aR,7aS)-4-[(4-fluorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-3-hydroxypropan-1-one
N-(furan-2-ylmethyl)-2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-methyl-4-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-1-(4-methylphenyl)piperazin-2-one
4-cyano-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-1H-pyrrole-2-carboxamide
N-cyclohexyl-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
3-({1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
2-[(4aR,7aS)-4-[(3-fluorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
4-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-1λ6-thiomorpholine-1,1-dione
6-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1,2-dihydropyridin-2-one
2-(2-oxo-1,2-dihydropyridin-1-yl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]acetamide
2-methyl-9-[2-(oxolan-2-ylmethoxy)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-4-(piperidin-1-ylmethyl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)benzamide
4,4,4-trifluoro-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]butan-1-one
4-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1,2-dihydrophthalazin-1-one
5-cyclopropanecarbonyl-1'-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-benzyl-4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,3-thiazole
(3S,5R)-N-benzyl-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carboxamide
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-methanesulfonylpiperidine
3-[(2-methyl-3-oxopiperazin-1-yl)methyl]-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
7-methyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide
4-(1H-pyrazol-1-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]benzene-1-sulfonamide