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N-[(8-methoxyquinolin-5-yl)methyl]-N-methylmorpholine-2-carboxamide
4-{1-[1-(4-methylbenzoyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
2-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3-methoxyphenol
11-{2-[2-(4-methylpiperidin-1-yl)-2-oxoethoxy]phenyl}-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
5-{2-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
2-butyl-4-methyl-3-oxo-N-[4-(pyridin-3-yloxy)phenyl]piperazine-1-carboxamide
N-(2-{5,6-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-2-yl}ethyl)imidazo[1,2-a]pyridine-6-carboxamide
2-{[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-6-methylpyridin-3-ol
2-methyl-5-{[3-(1,2-oxazolidine-2-carbonyl)-1,2-oxazol-5-yl]methoxy}-1,3-benzothiazole
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-(propan-2-yl)pyrimidin-4-amine
8-(2-methoxy-4-methylbenzenesulfonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1s,4s)-4-hydroxy-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)cyclohexane-1-carboxamide
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
2-[4-(2-methoxypyridin-3-yl)phenyl]-5-methylpyrimidine
8-(2,4-difluorobenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[4-(1-hydroxyethyl)phenyl]-1H-indazole-3-carboxylic acid
2-[({1-azabicyclo[2.2.2]octan-3-yl}amino)methyl]-4-(2H-1,3-benzodioxol-5-yl)phenol
(3R,4R)-1-{[3-(4-chlorophenoxy)phenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
5-(2-fluorophenyl)-2-(pyridin-3-yl)-4-[1-(thiophen-3-ylmethyl)piperidin-3-yl]pyrimidine
propan-2-yl 2-chloro-5-(4-oxopentanamido)benzoate
2-(1-benzylpiperidin-4-yl)-N-methylacetamide
3-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
2-[4-(2-methoxyethoxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
6-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
N-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-[2-(morpholin-4-yl)ethyl]piperazine-1-carboxamide
2-[2-({6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-3,4-dihydroquinazolin-4-one
2-[5-(3-hydroxyphenyl)-1H-indol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
methyl (2R)-2-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)propanoate
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(methyl)[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
ethyl 4-(2-phenylethyl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxylate
2-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}amine
2-(5-fluoro-2-methylphenyl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)acetamide
3-acetamido-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]benzamide
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}cyclopentan-1-ol
1-[benzyl(methyl)amino]-3-[4-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
6-fluoro-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
N3-benzyl-1-cyclopropyl-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-methyl-2-[4-(oxan-2-ylmethyl)phenoxy]acetamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(1-methyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
4-ethyl-3-[(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
6-(2,3-dihydro-1H-inden-1-ylmethyl)-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
(3R,5S)-N-(naphthalen-1-ylmethyl)-1-(propan-2-yl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
ethyl 4-[6-(2-cyclopropylquinoline-4-carbonyl)-6-azaspiro[2.5]octane-1-carbonyl]piperazine-1-carboxylate
6-[1-(4-chloro-2-fluorobenzoyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
1-(4-methyl-2-phenylpyrimidine-5-carbonyl)-3-propylpiperidine-3-carboxylic acid
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]propan-1-ol