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2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-[2-(pyridin-3-yloxy)propyl]acetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decane-3-carboxamide
9-[(5-ethylfuran-2-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-5-[4-(3-methoxypropyl)piperazine-1-carbonyl]pyrimidine
1-(3-methoxyphenyl)-4-[2-(1H-1,2,4-triazol-1-yl)propanoyl]piperazin-2-one
N,3-dimethyl-4-oxo-N-(pyridin-2-ylmethyl)-3,4-dihydrophthalazine-1-carboxamide
4-methyl-2-propyl-6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
4-[(4-fluorophenyl)methyl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine
N,N,4-trimethyl-3-{[(prop-2-en-1-yl)(propan-2-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-cyclopentanecarbonyl-N-(quinolin-2-ylmethyl)piperidine-4-carboxamide
(3S,4S)-4-methyl-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine-3,4-diol
N-[(4,6-dimethylpyridin-2-yl)methyl]-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
4-[1-(carbamoylmethyl)-3,5-dimethyl-1H-pyrazol-4-yl]-2-chlorobenzamide
N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-(pyrimidin-2-ylsulfanyl)acetamide
(2S)-2-amino-4-hydroxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}butanamide
N-(2-hydroxyethyl)-N,15-dimethyl-13-oxo-9-(thiophen-2-yl)-4-(trifluoromethyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
5-methyl-N-{4-[(quinolin-8-yl)carbamoyl]phenyl}furan-3-carboxamide
6-chloro-2-(1-ethyl-1H-pyrazol-4-yl)-N-methyl-N-propylquinoline-4-carboxamide
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-3-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1,4-dihydropyridin-4-one
4-(diphenylmethyl)-4-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[1-(3-chloro-2-fluorobenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
4-methyl-2-(propan-2-yl)-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-1,3-thiazole-5-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
8-[(2,2-difluoro-2H-1,3-benzodioxol-4-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
8-(1,3-benzothiazol-2-ylmethyl)-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(4-cyclopropyl-5-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
1-cyclopropyl-N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
[(1,4-dimethylpiperidin-4-yl)methyl][(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amine
1-[2-(dimethylamino)ethyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-oxopyrrolidine-3-carboxamide
2-(3-{3-cyclopropyl-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}phenoxy)acetamide
1-(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl)piperidin-4-ol
2-{4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-cyclohexylpiperazin-2-yl}ethan-1-ol
2-(dimethylamino)-2-(3-methylphenyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
1-{3-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(4-chloro-3-methylphenyl)-2-[4-(oxolan-2-ylmethyl)piperazin-1-yl]acetamide
N-[2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(phenylsulfanyl)acetamide
3-hexyl-1-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
[1-(2,6,8-trimethylquinoline-4-carbonyl)-2,5-dihydro-1H-pyrrol-2-yl]methanol
methyl 2-({2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazol-4-yl}formamido)acetate
4-cyclopentanecarbonyl-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(5-ethyl-1,3-oxazole-4-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 8-(2,3-dihydro-1-benzofuran-2-carbonyl)-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
(2R,3S,6R)-5-(isoquinoline-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-2-methoxypyridine-3-carbonitrile
(2S,4S)-1-benzyl-4-{[(2,3-dimethoxyphenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
(2H-1,3-benzodioxol-4-ylmethyl)[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
(3S,4S)-1-{2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-4-propylpyrrolidine-3-carboxylic acid
N,5-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrazine-2-carboxamide
3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1-(2-methyl-5-sulfamoylphenyl)urea