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2-benzyl-4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1,3-thiazole
1-(4-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-3,5-dimethyl-1H-pyrrol-2-yl)ethan-1-one
(3R,4R)-3-cyclobutyl-4-methyl-1-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}pyrrolidin-3-ol
2-[(3,5-difluorophenyl)methyl]-8-(1,3-thiazol-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
3-(carbamoylmethoxy)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]benzamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
2-(2-benzylmorpholine-4-carbonyl)-N,N-dimethylaniline
1-(3,5-dimethylphenyl)-4-[2-(3-hydroxyphenyl)acetyl]piperazin-2-one
[(5-{1-[(2,4-dimethylphenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
6-(6-methoxypyridin-3-yl)-N-(propan-2-yl)pyrimidin-4-amine
3-(2-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
2-amino-6-(4-hydroxyphenyl)-4-[4-methoxy-3-(methoxymethyl)phenyl]pyridine-3-carbonitrile
4-(2-chlorophenyl)thieno[2,3-d]pyrimidine
N-(1-cyclopentyl-1H-pyrazol-5-yl)azocane-1-carboxamide
1-ethyl-8-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(1-methylpiperidin-3-yl)ethyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
2-{[(2-methanesulfonylethyl)amino]methyl}-6-methylquinolin-4-ol
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]benzamide
4-[7-(3-methyl-1H-pyrazole-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]thiomorpholine
N-methyl-3-(1,2-oxazinan-2-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-phenyl-5-(thiomorpholine-4-sulfonyl)benzamide
4,6-dimethyl-1-(2-{[1-(2-methyl-1H-imidazol-1-yl)propan-2-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-2,3-dimethylbenzene-1-sulfonamide
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(quinolin-5-ylmethyl)acetamide
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(4-ethoxyphenyl)methyl]methylamine
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
1-(diphenylmethyl)-N-[(4-ethylphenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-[4-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)morpholin-3-yl]acetic acid
5-(2,4-difluorophenoxymethyl)-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-6-methylpyridine-2-carboxamide
2-(pyrrolidin-3-yl)-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]benzamide
(1S,5R)-6-[(1-methyl-1H-indol-2-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[4-(benzyloxy)phenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(2-methoxyethyl)-N-methyl-1H-pyrazole-4-carboxamide
N'1-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropane-1,1-dicarboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(6-methylquinolin-5-yl)methyl]pyrrolidin-3-yl]methanol
2,6-dimethyl-4-({[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]amino}methyl)phenyl acetate
(2R,3R,6R)-5-(1H-imidazol-2-ylmethyl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4,6-dimethyl-2-oxo-N-[1-(pyrazin-2-yl)propan-2-yl]-1,2-dihydropyridine-3-carboxamide
8-[(2S)-2-aminohexanoyl]-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(2R,6R)-4-(6-methoxyhexanoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2S,4R)-4-amino-N-methyl-1-{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}pyrrolidine-2-carboxamide
3-{2-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-2-oxoethyl}-4-(pyridin-3-ylmethyl)piperazin-2-one
4-methyl-N-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
N-methyl-5-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}butanamide
ethyl 2-({[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)acetate
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-(2-methyl-1H-indol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one