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1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(pyridin-4-yl)ethan-1-one
6-methyl-2-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}-1,3-benzothiazole
2-(4-{[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)pyrimidine
7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-4-(1H-pyrazol-3-yl)benzamide
methyl 1-[(3S,5S)-1-cycloheptyl-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(1-{1-[(2-methylphenyl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl}cyclopropyl)methanol
methyl 3-(furan-3-amido)-1-(2-methylpropyl)-5-({[4-(methylsulfanyl)phenyl]methyl}amino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-ethyl-5-methyl-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
1-{3-[4-(5,6-dimethylpyrimidin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
1-[2-methoxy-4-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
4-[(diethylamino)methyl]-5-ethyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}furan-2-carboxamide
(3S,4R)-1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-{3H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(1S,9aR)-1-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}-octahydro-1H-quinolizine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-[4-(propan-2-yl)piperazin-1-yl]pyridine-3-carboxamide
(1S,5R)-3-(2,5-difluorobenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(diphenylmethyl)-1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-1,2,3-triazole
4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1,3,5-trimethyl-1H-pyrazole
3-{1-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}benzoic acid
1-benzyl-5-(cyclopropylamino)-N-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2-(methoxymethyl)piperidine
1-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-3-[5-(2-methylphenyl)-1,3,4-thiadiazol-2-yl]urea
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
(2S)-2-amino-3,3-dimethyl-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]butan-1-one
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-methoxypyridine-3-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-(2-methoxyacetyl)-2,7-diazaspiro[4.5]decan-6-one
2-(quinolin-8-yl)benzonitrile
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-(2-phenoxyethyl)piperazine
3-{3-[1-(4,4,4-trifluorobutyl)-1H-pyrazol-3-yl]phenyl}pyridine
N3-(cyclopropylmethyl)-1-(2-methoxyethyl)-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-N3-propyl-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-4-propyl-6-[3-(pyridin-2-yl)azetidin-1-yl]pyrimidine
N-cyclopentyl-N-(3-phenylprop-2-yn-1-yl)-3-(pyrimidin-2-yloxy)benzamide
4-{5-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrimidin-2-yl}morpholine
3-(4-chlorophenyl)-4-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}butanoic acid
2-cyclopropyl-N-(2,4-dimethylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propan-1-one
1-[2-(2,5,7-trimethyl-1H-indol-3-yl)acetamido]cycloheptane-1-carboxamide
(4aR,7aS)-1-methyl-4-(2,5,7-trimethylquinoline-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-butyl-N-[2-(morpholin-4-ylmethyl)phenyl]-2,5-dihydro-1H-pyrrole-1-carboxamide
5-[1-(2-methylpropyl)pyrrolidin-2-yl]-N-(1H-pyrazol-3-yl)thiophene-2-carboxamide
[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl](methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-(2,6-dimethoxypyridine-3-carbonyl)-4-(2,6-dimethylpyridin-4-yl)piperazine
6-cyclopentyl-N,1-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[3-(2-{4-[3-(3-fluorophenyl)benzoyl]piperazin-1-yl}ethoxy)phenyl]methyl}morpholine
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(carbamoylmethyl)acetamide
(1S,5R)-6-(cyclopropylmethyl)-3-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
2-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]pyridine-4-carboxamide