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8-benzyl-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(2-ethyl-1H-imidazol-1-yl)-N-[(1-methylpiperidin-3-yl)methyl]acetamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine
6-chloro-N,N-dimethyl-3-[({[2-(trifluoromethoxy)phenyl]methyl}amino)methyl]imidazo[1,2-a]pyridine-2-carboxamide
6-{1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-4-yl}pyrimidin-4-ol
4-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-1-(3-methoxyphenyl)piperazin-2-one
1-(cyclopropylmethyl)-4-(2-methylpyridine-3-carbonyl)-2-(propan-2-yl)-1,4-diazepane
methyl({[5-(oxan-2-yl)thiophen-2-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
3-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-1-phenylpyrrolidin-2-one
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridine
4-(1H-imidazol-1-ylmethyl)-1-{[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}piperidin-4-ol
3-(2-ethyl-1H-imidazol-1-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]propanamide
methyl 2-(morpholine-4-sulfonyl)-6-(2-phenylpropyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-3-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(2-fluorophenoxymethyl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrazole-3-carboxamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
3-{2-oxo-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethyl}-4-(thiophen-2-ylmethyl)piperazin-2-one
N-butyl-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carboxamide
4-ethyl-3-{1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[6-(pyrrolidin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}cycloheptanamine
methyl (2R)-2-(3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamido)propanoate
2-methyl-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-1,3-benzoxazole-6-carboxamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-(3-cyanopyridin-2-yl)-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
{2-[(4-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)methyl]phenyl}methanol
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)[(6-methylpyridin-2-yl)methyl]amine
1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-(1-benzoylpiperidin-4-yl)-N-cyclopropylpiperidine-3-carboxamide
5-(2-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}ethyl)-1,3,4-thiadiazol-2-amine
8-methoxy-3-[(2R)-pyrrolidin-2-ylmethyl]-3,4-dihydroquinazolin-4-one
(3S,5S)-5-[(4-fluorophenyl)carbamoyl]-1-[(4-methoxyphenyl)methyl]piperidine-3-carboxylic acid
1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-6-methylimidazo[1,2-a]pyridine-2-carboxamide
3-(3-methoxyphenyl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
[3-(1H-1,2,3-benzotriazol-1-yl)propyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
1-(1-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-1,8-naphthyridine
3-(3-methoxyphenyl)-6-(1H-pyrazole-4-carbonyl)-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[2-(dimethylsulfamoyl)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[(4-fluorophenyl)methyl]-4-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2-(propan-2-yl)-1,4-diazepane
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(2,2-dimethylpropyl)piperazin-2-yl]ethan-1-ol
1-{1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
2-{2-[(2-ethyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]phenoxy}acetic acid
1-(3-cyclopentylpropyl)-3-(pyrrolidin-1-yl)piperidine
4-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-4-oxobutanamide
6-[(oxan-4-yl)amino]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
N-{[3-methyl-7-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-[(4-hydroxyphenyl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one