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1-acetyl-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-4-carboxamide
N,N-diethyl-5-methyl-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
dimethyl[(1-{[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]amine
2,2-dimethyl-N-(1-{1-[2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
N-(2-fluorophenyl)-3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
(2S,4S)-4-amino-1-{3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propanoyl}-N-ethylpyrrolidine-2-carboxamide
3-({1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
(2Z)-2-fluoro-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-phenylprop-2-en-1-one
[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)pyrrolidin-3-yl]methanamine
2-cyclobutyl-N-[(3R,4S)-4-propyl-1-(pyrimidin-2-yl)pyrrolidin-3-yl]acetamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
4-(5-{[(3-fluorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)-N-(prop-2-en-1-yl)piperidine-1-carboxamide
{1-[1-(2,2-diphenylethyl)piperidin-3-yl]piperidin-4-yl}methanol
1-cyclohexyl-5-{3-[2-(dimethylamino)ethyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-(4-methyl-2-phenyl-1H-imidazol-1-yl)acetamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(6-methylpyridin-2-yl)methyl]acetamide
N-[(3S,5S)-1-(2-ethoxyacetyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[(4-chlorophenyl)methyl]-5-(3-methoxypiperidine-1-carbonyl)-1,3-benzoxazole
(1R,5S)-6-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}-6-azabicyclo[3.2.1]octane
5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-1H-indazole
2-(4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-1H-pyrazol-5-amine
3-{2-oxo-2-[(2S)-2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethyl}imidazolidine-2,4-dione
N-ethyl-N-(2-hydroxyethyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(3-chlorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]pyridine-4-carboxamide
2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)acetamide
8-(2-ethylpyridine-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-4-methyl-2-(propan-2-yl)pyrimidine-5-carboxamide
9-[(2S)-2-amino-3-hydroxypropanoyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-ethyl-2,3-dimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
ethyl 1-(3-methylbutyl)-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-{1-[5-(methylcarbamoyl)furan-2-yl]-1H-imidazol-2-yl}benzoic acid
2-(2,3-difluorophenyl)-1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
7-(2-methylphenyl)-4-(1,3-thiazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-methyl-3-[4-(4H-1,2,4-triazol-4-ylmethyl)phenyl]-1,2,4-oxadiazole
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
N-[(7-chloro-4-{[(4-fluorophenyl)methyl]amino}quinazolin-2-yl)methyl]-2-(methylsulfanyl)benzamide
N-[(1R,3S)-3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]cyclopentyl]-2,5-dimethyl-1,3-oxazole-4-carboxamide
3-({[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amino}methyl)-N-methylpyridin-2-amine
2-{5-[3-(cyclopentylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]thiophen-2-yl}-1H-imidazole
(3S,7S)-5-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
1-{4-[(1-hydroxy-3-methylbutan-2-yl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
4-[4-(3-methoxypropyl)piperazine-1-carbonyl]-6-methyl-1,2-dihydroquinolin-2-one
1-(4-{4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}-1,4-diazepan-1-yl)ethan-1-one
(4aR,8aS)-6-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-[(3,4,5-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
1-[4-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-[(3S,4R)-4-(propan-2-yl)-1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]pyrrolidin-3-yl]methanesulfonamide
3-[(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)methyl]benzoic acid