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1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}azepane
(3aS,7aR)-5-methyl-2-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
3-methyl-5-[4-(pyrrolidin-1-ylmethyl)phenyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
methyl({[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})(thiophen-3-ylmethyl)amine
5-[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-4-yl]-5-propylimidazolidine-2,4-dione
2-{4-[4-(ethylamino)pyrimidin-2-yl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(1-ethylpiperidin-3-yl)methyl]-3,4-dimethoxybenzamide
3-(pyrimidin-5-yl)-4H-chromen-4-one
N-(2-hydroxyethyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
(3R,4R)-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
1-[(4-methylphenyl)methyl]-4-(pyrrolidin-3-ylmethyl)piperazin-2-one
2-[(3,4-difluorophenyl)methyl]-8-(2-methoxyacetyl)-2,8-diazaspiro[4.5]decan-3-one
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[3-(methylsulfanyl)propyl]benzamide
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(furan-2-ylmethyl)(prop-2-yn-1-yl)amine
(3R,4R)-4-amino-1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-3-ol
6-(cyclohex-3-en-1-ylmethyl)-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-methoxyphenyl)propanamide
2,3,5-trimethyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
{[2-(cyclopentyloxy)phenyl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-2-(4-fluorophenyl)-N-(pyridin-3-ylmethyl)acetamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-oxo-2-(thiophen-2-yl)acetamide
4-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-2-[2-(2-methoxyethyl)-2H-1,2,3,4-tetrazol-5-yl]morpholine
N-(1,4-dioxan-2-ylmethyl)-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-{1-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-phenoxyacetamide
2-(3-oxo-9-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-2-yl)propanoic acid
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-(cyclopropylmethyl)piperazine
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2,3-dihydro-1-benzofuran-5-carboxamide
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-methyl-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-7-methyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
N-[2-(4-methoxyphenyl)phenyl]-1-(3-methoxypropanoyl)pyrrolidine-2-carboxamide
2-(dimethylamino)-N-[2-(dimethylsulfamoyl)ethyl]-2-(3-fluorophenyl)acetamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
6-amino-2-(2-{[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]amino}ethyl)pyrimidin-4-ol
N-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-3-yl]methyl}-1H-indazole-3-carboxamide
2-ethyl-N-[2-(2-methylpropanesulfonyl)ethyl]pyrimidine-5-carboxamide
4-[2-(piperidine-1-carbonyl)phenoxy]-1-{[4-(propan-2-yloxy)phenyl]methyl}piperidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(2-oxopyrrolidin-1-yl)propanamide
8-benzyl-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-N-cyclopentylfuran-2-carboxamide
4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-(2-phenylethyl)piperidine
(4aS,7aR)-4-cyclobutanecarbonyl-N-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl][(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl](pyridin-3-ylmethyl)amine
(2R,6R)-4-[(1,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-6-carboxylic acid
2-chloro-5-[3-(1-methoxyethyl)phenyl]-N-methylbenzamide
N-[1-(6-methyl-2-phenylpyrimidin-4-yl)pyrrolidin-3-yl]acetamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide
(2S,4S)-1-cyclopentyl-N-ethyl-4-[4-(1H-imidazol-1-yl)butanamido]pyrrolidine-2-carboxamide