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N-[(3S,4R)-1-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-4-propylpyrrolidin-3-yl]acetamide
1-cyclobutanecarbonyl-4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyridine-3-carboxamide
N3-methyl-N3-(2-methylpropyl)-4-oxo-N5-(2-phenylethyl)-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclobutanecarboxamide
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-5-(methoxymethyl)furan-2-carboxamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]acetamide
3-[(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)oxy]pyridine
8-(4-hydroxy-3,5-dimethylphenyl)-2-(morpholin-4-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-{2-[7-(3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclobutanecarboxamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
(4aS,8aR)-6-(1-benzofuran-5-carbonyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-(2-hydroxypropyl)-6-(4-methoxyphenyl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(2-methoxyethyl)-8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{1-[3-(cyclohexyloxy)-2-hydroxypropyl]-1H-imidazol-2-yl}phenol
N-[1-({[3-(pyridin-3-yloxy)propyl]carbamoyl}methyl)-1H-pyrazol-4-yl]furan-2-carboxamide
4-[2-(2-chloro-3,4-dimethoxyphenyl)-1H-imidazol-1-yl]-1-methylpiperidine
1-(adamantan-2-yl)-4-[(2S,4S)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carbonyl]piperazine
2-[9-(2,4-difluorobenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
1-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
3-{1-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-5-methyl-4H-1,2,4-triazole
7-[(2S)-2-amino-6-hydroxyhexanoyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1S,5R)-6-benzyl-3-(2,5-dimethylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(4-carbamoylpyridin-2-yl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
N-(1,4-dimethyl-1H-pyrazol-5-yl)-2-(1-methylpiperidin-2-yl)acetamide
1-(4-methyl-1,3-thiazol-2-yl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-(2-methoxy-2-methylpropyl)-3,6,7-trimethyl-1-benzofuran-2-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-(1-methylpiperidine-4-carbonyl)morpholine
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-N-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-5-carboxamide
3-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1-[5-(2-phenylethyl)-1,3,4-thiadiazol-2-yl]urea
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(2-hydroxy-2-phenylethyl)-N-methylacetamide
3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-phenyl-4-[(1s,4s)-4-aminocyclohexyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[4-(4-methoxypyrimidin-2-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(thiophen-2-yl)butan-1-one
N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
(3S,4S)-4-{[(4,6-dimethylpyridin-2-yl)methyl](methyl)amino}-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-ol
2-(pyridin-3-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-(2-amino-4-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}-6-methylpyrimidin-5-yl)propanoic acid
ethyl 3-{[1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
3-{1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
4-{4-[2-(3-fluorophenyl)acetamido]-1H-pyrazol-1-yl}-N-[2-(1H-indol-3-yl)ethyl]benzamide
2,3-dimethyl-6-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
4-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}phenol