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N-(2,4-difluorophenyl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-methyl-1-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]urea
1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-5-(thiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{[5-(2-methylpropyl)-4-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-[(2R,3R,6R)-5-(3-fluoro-4-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[1-({[(3S)-2-oxoazepan-3-yl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
N-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-[4-(4-fluorophenoxy)piperidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
N-[(1S,2R)-2-aminocyclobutyl]-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-(pyridin-3-yl)-7-(pyrrolidine-1-sulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-{[(1,3-benzoxazol-2-ylmethyl)(methyl)amino]methyl}-N-phenyl-1,3-thiazol-2-amine
2-(4-methylpentyl)-4-(1H-pyrazole-4-carbonyl)morpholine
N-ethyl-1-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
methyl (2S,3S)-2-{[5-(butylcarbamoyl)-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridin-3-yl]formamido}-3-methylpentanoate
N-(1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
N-(2-hydroxyethyl)-1-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-indole-6-carboxamide
2-[1-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-(1-methylpiperidin-4-yl)formamido]acetic acid
(1S,3R)-3-{[(2H-1,3-benzodioxol-5-yl)carbamoyl]amino}-N-(4-fluorophenyl)cyclopentane-1-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-2-(methylamino)pyridine-4-carboxamide
2-(3-phenylpiperidin-1-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}acetamide
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[4-(4-methoxyphenyl)butan-2-yl]-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
5-[(1,3-benzothiazol-2-ylmethyl)(methyl)amino]-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-ethyl-3-[1-(5-phenylpentanoyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-methyl-4-{[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(1-{2-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-2-yl)methanol
4-chloro-N,N-dimethyl-5-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}-1,3-thiazol-2-amine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(furan-3-ylmethyl)-N-methyl-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
2-amino-7-methyl-4-(1-phenyl-1H-pyrazol-5-yl)-5H,7H-furo[3,4-b]pyridine-3-carbonitrile
(1R,5S)-3-[(4-methanesulfonylphenyl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonane
(3R,4S)-4-cyclopropyl-1-[4-(1H-imidazol-1-yl)benzoyl]pyrrolidin-3-amine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxamide
benzyl 3-{[(5-acetyl-4-methylpyrimidin-2-yl)amino]methyl}piperidine-1-carboxylate
3-methyl-1-(2-methylpropyl)-4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-one
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})amine
3-[({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)methyl]pyrrolidin-3-ol
N-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(2,6-dimethylpyridin-4-yl)-4-(1-methyl-1H-pyrrole-2-carbonyl)piperazine
methyl 3-acetamido-5-[(furan-3-ylmethyl)amino]-1-[2-(1H-indol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(4-fluoro-2-methylphenyl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[2-(2-methoxyphenyl)ethyl]pyrrolidin-2-one
N-[(3R,4S)-1-[(5-chlorothiophen-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-hydroxyacetamide
[(4-{1-[(3,4-dimethoxypyridin-2-yl)methyl]piperidin-2-yl}phenyl)methyl]dimethylamine
3-(1H-1,2,3-benzotriazol-1-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]propanamide
N-[(1R,3R)-3-aminocyclopentyl]-2-[cyclohexyl(methyl)amino]pyridine-3-carboxamide
N-cyclopropyl-2-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)propanamide
4-methyl-3-[5-(3-methyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]pyridine
4,6-dimethoxy-2-[3-(pyridin-2-yl)azetidin-1-yl]pyrimidine
6-(2,5-dimethylfuran-3-yl)-2-(4-fluoropiperidine-1-carbonyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-{[4-(methylsulfanyl)phenyl]methyl}piperazine