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[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
1-ethyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H-pyrazole-5-sulfonamide
N-methyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(propan-2-yl)acetamide
5-({[(3-{2-[4-(2-ethylbutanoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
8-[2-(2,3-difluorophenyl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-cyclohexyl-3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propanamide
(3S)-4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
1-methyl-5-[3-(1H-pyrazol-1-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(1H-1,3-benzodiazol-5-yl)-3-(2-propoxyethyl)urea
3-{[(furan-3-ylmethyl)(methyl)amino]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
N-ethyl-4-methanesulfonyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
3-hydroxy-3-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)benzamide
1-(4-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-{1,3-dioxo-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
5-{[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]methyl}-N,N-dimethylfuran-2-carboxamide
dimethyl({2-[3-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)phenoxy]ethyl})amine
1-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}propanamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-N-(2-methoxyphenyl)piperidine-1-carboxamide
1-methyl-2-oxo-8-(2-propyl-1,3-thiazole-4-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
4-[4-({[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amino}methyl)phenyl]but-3-yn-1-ol
5,8-dimethyl-2-{[4-(oxolane-2-carbonyl)piperazin-1-yl]methyl}quinolin-4-ol
7-(1,3-benzothiazol-2-yl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-amino-6-hydroxypyrimidin-4-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
3-(2H-1,3-benzodioxol-5-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
N,N-dimethyl-2-[(1S,5R)-6-[(phenylcarbamoyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
1-[(5-acetylthiophen-3-yl)methyl]-4-phenylpiperidine-4-carbonitrile
(4aR,7aS)-1-methyl-4-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(oxan-4-yl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(2-methyl-7-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl)pyrrolidine
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2,2-dimethylcyclopropane-1-carboxamide
4-(1,3-dimethyl-1H-pyrazol-5-yl)-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4H-1,2,4-triazole
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-4-hydroxy-3-methylbenzamide
2-{4-[5-(furan-2-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl]piperazin-1-yl}ethan-1-ol
4-[2-(3-hydroxyphenyl)-1H-imidazol-1-yl]-N-phenylpiperidine-1-carboxamide
1-[(4-ethoxyphenyl)methyl]-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-{2-[(6-methoxypyrimidin-4-yl)amino]ethyl}pyridine-4-carboxamide
7-(2,2-diphenylethyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
7-(5-methylthiophen-2-yl)-4-(morpholine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamide
2-(dimethylamino)-N-[2-(ethylsulfanyl)ethyl]-4-methylpyrimidine-5-carboxamide
N-[(2-methylphenyl)methyl]-2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}-N-(prop-2-en-1-yl)acetamide
1-methyl-4-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
2-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}cyclopentanamine
2-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-N,N-dimethylaniline
(1S,5R)-3-[(4-methoxypyridin-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one