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N-cyclopropyl-2-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]acetamide
4-(2-methoxyphenyl)-N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)piperazine-1-carboxamide
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylpyridine-2-carboxamide
ethyl 1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4-(2-phenylethyl)piperidine-4-carboxylate
3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)-N-(5-methylpyridin-3-yl)benzamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
2-(2-methoxyphenyl)-5-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}pyrimidine
5-(1-{2-[1-(propan-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)-1H-indole
4-(2-methoxyphenyl)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
N-(2-methoxyethyl)-3-{[1-(thiolan-3-yl)piperidin-4-yl]oxy}benzamide
8-[(3,5-difluorophenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(dimethyl-1,3-oxazole-5-carbonyl)piperidin-3-ol
1-[2-({[1-(2-fluorophenyl)cyclopentyl]methyl}amino)-4-methylpyrimidin-5-yl]ethan-1-one
(1S,5R)-3-(1-methyl-1H-pyrrole-2-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(1-methyl-1H-pyrrol-2-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1H-pyrazole-5-carboxamide
N,1-dimethyl-6-propyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-3-(2-oxopyrrolidin-1-yl)benzamide
6-methyl-5-{5-[2-(thiophen-2-yl)ethyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
3-(3-chlorophenyl)-1-[(2,4,6-trimethoxyphenyl)methyl]pyrrolidine
3-(1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)propan-1-ol
N-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}-4-(pyridin-4-yl)piperazine-1-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2,5,7-tetramethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetyl)-N-ethylpyrrolidine-3-carboxamide
3-(4-chlorophenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-phenylpropanamide
2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pyridine-4-carboxamide
N-{3-[(1-hydroxybutan-2-yl)(pyridin-2-ylmethyl)carbamoyl]-2-methylphenyl}furan-2-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(6-methylpyridin-3-yl)ethyl]benzamide
1-[1-(2-phenoxyacetyl)piperidin-3-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-fluoro-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-5-sulfamoylbenzamide
2-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]thieno[2,3-d]pyrimidin-4-amine
1-[2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-oxoethyl]pyrrolidin-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)butanamide
(2S,4S)-1-(cyclohexylmethyl)-N-ethyl-4-(4-methylbenzamido)pyrrolidine-2-carboxamide
1-ethyl-4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-2-propyl-1,3-thiazole-4-carboxamide
2-(4-fluorophenyl)-4-[1-(methoxymethyl)cyclobutanecarbonyl]morpholine
2-(3-fluorophenoxymethyl)-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1,3-oxazole-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(1,1-dioxo-1λ6-thiolan-3-yl)piperidine-4-carboxamide
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[(3R,4R)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
6-tert-butyl-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(5-acetylthiophen-3-yl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
1-[3-({[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]ethan-1-one
methyl 2-(4-acetyl-4-phenylpiperidin-1-yl)propanoate
2-(3-hydroxypiperidin-1-yl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}acetamide
1-cyclopentyl-5-oxo-N-[2-(pyridin-3-yl)ethyl]pyrrolidine-3-carboxamide
5-methyl-6-(2-methylpiperidine-1-carbonyl)-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidin-4-amine
N-(2,3-dihydro-1H-inden-2-yl)-3-propyl-1H-pyrazole-5-carboxamide
dimethyl({[(3S,4R)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
2-[(4S)-4-hydroxy-3,3,4-trimethylpiperidine-1-carbonyl]-6-methyl-4H-pyran-4-one