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N-methyl-N-(2-phenylethyl)-2-(piperazine-1-carbonyl)-2,3-dihydro-1H-inden-2-amine
N,2-dicyclopentyl-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)acetamide
7-chloro-4-[2-methyl-6-(1-methylpiperidin-4-yl)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-[3-(dimethylamino)pyrrolidin-1-yl]-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
ethyl 4-(1-{[3-(furan-2-yl)phenyl]methyl}piperidin-3-yl)piperazine-1-carboxylate
1-({3-[4-methoxy-4-(prop-2-en-1-yl)piperidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-1,3-benzodiazole
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-4-yl]piperidin-3-ol
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-4-(hydroxymethyl)pyridine-2-carboxamide
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3-(methylsulfanyl)propanamide
(3-methylbutyl)({[1-(morpholin-4-yl)cycloheptyl]methyl})amine
1-[(2,4-difluorophenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-1-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-(pyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(cyclohexylmethyl)-1-(1H-indol-2-ylmethyl)-1,4-diazepan-5-one
[(2R)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]pyrrolidin-2-yl]methanol
2-{2-[2-(morpholin-4-ylmethyl)phenyl]phenoxy}propanamide
2-[5-(5-methyl-2H-1,2,3-triazol-4-yl)-1-[(4-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
1-(cyclohexylmethyl)-6-oxo-N-{3-[(pyridin-3-yl)amino]propyl}piperidine-3-carboxamide
(1R,5R)-N,N-dimethyl-6-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
N-[(2R,4R,6S)-2-cyclohexyl-6-(pyridin-4-yl)oxan-4-yl]benzamide
ethyl 4-(2-phenylethyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine-4-carboxylate
8-[(2-phenylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-({[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)pyrrolidin-3-ol
N-[3-(1H-indol-2-yl)phenyl]-1-(1-methylcyclopropanecarbonyl)piperidine-4-carboxamide
(1S,6R)-9-{[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
2-ethyl-6-{imidazo[1,2-a]pyridine-3-carbonyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N2-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
(3S,4S)-1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(piperidin-1-yl)pyrrolidin-3-ol
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(morpholin-4-yl)propan-1-one
4-(2,4-difluorophenoxy)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-4-carboxylic acid
4-methyl-2-propyl-6-[3-(pyridin-3-yl)azetidin-1-yl]pyrimidine
8-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-{[2-(dimethylamino)-2,3-dihydro-1H-inden-2-yl]formamido}propanamide
methyl({[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})(pyrazin-2-ylmethyl)amine
5-{pyrazolo[1,5-a]pyridin-7-yl}pyrazin-2-amine
3-{2-[2-(furan-2-yl)phenyl]-1H-imidazol-1-yl}-N-methylbenzamide
1-{2-[(benzylsulfamoyl)amino]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-one
2-{[5-(3-chloro-4-methoxyphenyl)-4-(4-methylphenyl)pyrimidin-2-yl]amino}acetamide
[(1R)-1-(3-methoxyphenyl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-[2-(diethylamino)ethyl]-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(quinolin-4-yl)piperidin-3-yl]propan-1-ol
2-benzyl-8-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(2-{[(1S)-1-phenylethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-cyclopropyl-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
1-{[3,5-dichloro-4-(propan-2-yloxy)phenyl]methyl}-N,N-dimethylazepan-4-amine
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(3-fluorophenyl)methyl]urea
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(6-fluoroquinolin-2-yl)methyl]pyrrolidin-3-yl]methanol