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2-(4-{[2-(5-methylfuran-2-yl)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
[(3-methoxyphenyl)methyl](methyl){[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
N-methyl-N-[(5-{7-oxo-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-5-yl}furan-2-yl)methyl]methanesulfonamide
2-(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyridine-3-carbonitrile
N-[1-(1H-indol-5-yl)ethyl]-3-(2-oxopiperidin-1-yl)propanamide
6-oxo-N-[(1-phenylcyclopentyl)methyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(2-methoxyethoxy)ethan-1-one
4-(1-{imidazo[1,2-a]pyridin-2-ylmethyl}-1H-imidazol-2-yl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}acetamide
1-(1H-imidazol-1-ylmethyl)-N-[2-methyl-4-(5-methyl-1,3-benzoxazol-2-yl)phenyl]cyclopropane-1-carboxamide
4-methyl-5-{[4-(2-phenylethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]pent-4-enamide
6-(dimethylamino)-N-[(2S)-oxolan-2-ylmethyl]pyridine-3-carboxamide
N-[2-(1H-imidazol-1-yl)propyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-yl)piperazine
(2S,4R)-4-amino-N,N-diethyl-1-(2-methanesulfonylacetyl)pyrrolidine-2-carboxamide
1-(difluoromethyl)-4-(5-fluoro-2-methoxyphenyl)-5-methyl-1H-pyrazole
(2R,3S,6R)-3-(4-methylphenyl)-5-(pyridin-3-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-tert-butyl-6-oxo-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
5-methyl-N-{[5-(methylsulfanyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]methyl}thiophene-2-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-2-one
8-[(1R,2R,3S,4S)-3-aminobicyclo[2.2.1]heptane-2-carbonyl]-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
3-[2-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)carbamoyl}amino)phenyl]-N-methylpropanamide
N-cyclooctyl-1-(2-methoxyethyl)-5-(2-methylpiperidine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-methyl-1-[4-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)piperidin-1-yl]butan-1-one
methyl 3-({[(2-hydroxyadamantan-2-yl)methyl]carbamoyl}amino)-4-methoxybenzoate
3-[(dimethylamino)methyl]-1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
2-cyclopropyl-5-[1-(2,4-difluorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]pyrimidine
1-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2S,4R)-4-amino-N-(propan-2-yl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidine-2-carboxamide
3-methyl-7-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-[3-(3-methoxyphenyl)phenyl]-N-(pyridin-3-ylmethyl)piperidin-4-amine
N-(carbamoylmethyl)-2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-[1-(7-{[3-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-3-methylbutyl]pyridine-3-carboxamide
dimethyl({[5-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)thiophen-3-yl]methyl})amine
3-{3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2-methoxypyridine
1-[(2-chlorophenyl)methyl]-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
7-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[(3-{8-methyl-2,8-diazaspiro[5.5]undecane-2-carbonyl}-1,2-oxazol-5-yl)methyl]piperidin-4-ol
3-{2-amino-4-methyl-6-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]pyrimidin-5-yl}propanoic acid
N-[(5-methylthiophen-2-yl)methyl]-1,1-dioxo-N-(pyridin-4-ylmethyl)-1λ6-thiolane-3-carboxamide
N-[3-(4-methoxyphenyl)propyl]-6-[4-(methylamino)piperidin-1-yl]pyridine-3-carboxamide
3-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}-N-(1,3-thiazol-2-yl)propanamide
2-(1-methyl-1H-indol-3-yl)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}thiomorpholine
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[(1r,4r)-4-hydroxycyclohexyl]propanamide