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3-(4-chlorophenyl)-1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]propan-1-one
1-methyl-5-[({5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)methyl]pyrrolidin-2-one
3,5-dimethoxy-2-{[methyl(oxan-4-yl)amino]methyl}benzoic acid
4-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]morpholine
2-(2-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
4-[(3-{1-[(3-fluorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]morpholine
8-(3-acetyl-1H-pyrazole-5-carbonyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(4-cyanophenyl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
5-chloro-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
(2S,4R)-4-amino-N,N-diethyl-1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]pyrrolidine-2-carboxamide
methyl 4-{[(2-{1-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
N-{4-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]phenyl}methanesulfonamide
1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-(pyrrolidine-1-carbonyl)piperidine
(3aS,6aS)-2-methyl-5-[(2,4,5-trimethoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(4-chlorophenyl)-5-(propane-1-sulfonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[(1-methylpiperidin-3-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
4-({5-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
1-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-(1-{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-yl)ethan-1-ol
5-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-3,4-dihydropyrimidin-4-one
methyl 1-(9-methoxy-7-oxo-3-{[4-(propan-2-yl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl)piperidine-2-carboxylate
N-benzyl-4,6-dimethyl-2-oxo-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(prop-2-en-1-yl)acetamide
methyl 4-({3-[2-(dimethylamino)ethyl]-1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)benzoate
N-(3-hydroxy-3-methylbutyl)-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
8-[(3-hydroxyphenyl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
dimethyl(3-{2-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(2-methylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-ethyl-5-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-cyano-N,1-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-1H-pyrrole-2-carboxamide
N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2,5-dimethoxy-N-[2-(1-methylpiperidin-3-yl)ethyl]benzamide
4-({5-[1-(2H-1,3-benzodioxol-5-yloxy)ethyl]-1-ethyl-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
3-(2-propoxypropyl)-1-(2,3,4-trifluorophenyl)urea
2-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]pyrrolidin-2-yl}-1,3-benzothiazole
N5-ethyl-N5-[2-(1H-pyrazol-1-yl)ethyl]-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[(6-methylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazine-1-carboxylate
N-({1-[(3-fluoropyridin-4-yl)methyl]piperidin-4-yl}methyl)-5-hydroxypyrazine-2-carboxamide
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-3-phenylpropan-1-one
1-[(2R,3R)-2-hydroxy-3-(1,2,3,6-tetrahydropyridin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(methylsulfanyl)ethan-1-one
(4aS,8aS)-2-[(2,6-difluoro-3-methoxyphenyl)methyl]-decahydroisoquinolin-4a-ol
2,8-dimethyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}quinoline-4-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-[4-(propan-2-yl)phenyl]acetamide
1-(4-{2-[4-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
4-(3-{[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]amino}propyl)piperazin-2-one
(4aS,7aR)-1-[2-(methylamino)acetyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide