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1-(3-fluoro-4-methoxybenzoyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
N-[(3,4-dichlorophenyl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
3-chloro-4-{[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]oxy}-N-cyclopentylbenzamide
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-imidazol-1-yl)ethan-1-one
1-(4-{2-[(5-chloropyrimidin-2-yl)oxy]hex-5-en-1-yl}piperazin-1-yl)ethan-1-one
2-[methyl(oxan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-(2-chlorophenyl)-3-[1-(1-cyclopentylpiperidin-4-yl)-1H-pyrazol-5-yl]urea
2-(2,3-difluorophenyl)-1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
6-[1-(azepan-1-yl)-1-oxopropan-2-yl]-5,6-dihydro-1,6-naphthyridin-5-one
6-[methyl(oxan-4-yl)amino]-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
1-[(1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
6-(4-fluorophenyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N,3,4,7-tetramethyl-N-(quinoxalin-2-ylmethyl)-1H-indole-2-carboxamide
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
({5-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-yl]methanol
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[(1-phenylcyclohexyl)methyl]propanamide
3-{4-phenyl-5-[4-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}propanamide
3-({[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)propane-1,2-diol
2-[5-(2-methyl-1-benzofuran-5-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
(2R,6S)-4-[1-(3-methoxypyrazin-2-yl)piperidin-4-yl]-2,6-dimethylmorpholine
2-[(1S,5R)-6-(2,1,3-benzothiadiazol-5-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-2,6-dimethylquinoline
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-[2-(trifluoromethyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-chloro-4-({[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenol
4-{4-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]piperidine-1-carbonyl}pyridine
3-cyclopentyl-5-(2-methyl-1,3-thiazol-4-yl)-1-{[1,2,4]triazolo[4,3-b]pyridazin-6-yl}-1H-1,2,4-triazole
3-(1H-pyrazol-1-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
{9-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(1H-imidazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
(3S,4S)-1-(3,5-dichlorobenzoyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
N-(adamantan-2-ylmethyl)-6-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
N-({1-[(3,5-dimethyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)-3-methylbut-2-enamide
(1R,5R)-6-(cyclobutylmethyl)-3-(4-methanesulfonylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N,N-dimethyl-2-({1-[(1-methyl-1H-pyrrol-2-yl)methyl]piperidin-4-yl}formamido)propanamide
(1S,5S)-3-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
6-chloro-4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methylquinoline
4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}thiomorpholine
(3R,4R)-1-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-ol
2-amino-4-{2-phenylimidazo[1,2-a]pyrimidin-3-yl}-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl})(propan-2-yl)amine
N-[2-(diethylamino)ethyl]-N-ethyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-yl)benzoic acid
1-(azepan-1-yl)-3-[4-chloro-2-(1,2-oxazinan-2-ylmethyl)phenoxy]propan-2-ol
1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)-3-(1H-pyrazol-5-yl)piperidine
6-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]quinoxaline
2-cyclopropyl-8-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
[2-({4-[(3,4-difluorophenyl)methyl]piperazin-1-yl}methyl)phenyl]methanol
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-{[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile