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1-propyl-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
{5-[(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)methyl]furan-2-yl}methanol
1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-N-[2-(1H-imidazol-4-yl)ethyl]piperidin-4-amine
5-[5-(butan-2-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-(oxolane-3-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N-(1-benzothiophen-5-ylmethyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-methoxy-4-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenol
1-{1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazole-4-carbonyl}azocane
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]acetamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(2,3-dihydro-1H-indol-1-yl)ethan-1-one
N-[2-(2-methyl-1H-indol-3-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
3-(2-methoxyethyl)-1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperidine-3-carboxylic acid
[(4-fluorophenyl)methyl][(2E)-2-methylbut-2-en-1-yl](pyridin-4-ylmethyl)amine
8-[(3-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1,2-oxazol-5-yl)methoxy]quinoline
3-({2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}methyl)-5-(oxolan-2-yl)-1,2,4-oxadiazole
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
(4aS,7aR)-4-benzyl-N-ethyl-N-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-sulfonamide
7-cyclohexyl-2-(3-hydroxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
1-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}benzoyl)pyrrolidine
[4-benzyl-1-(2,3-dimethyl-1H-indole-5-carbonyl)piperidin-4-yl]methanol
1-methyl-N-[1-(thiophen-2-yl)propan-2-yl]-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
9-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
8-(1,3-benzothiazol-2-ylmethyl)-1-benzyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-fluoro-4-[2-(4-fluorophenyl)azetidine-1-carbonyl]-2-methylquinoline
2-{2-chloro-4-[(4,4-difluoropiperidin-1-yl)methyl]-6-methoxyphenoxy}acetic acid
5-(2-fluorophenyl)-N-[(4-phenyloxan-4-yl)methyl]-1,2,4-triazin-3-amine
1-[(ethylcarbamoyl)methyl]-N-[3-(3-methoxyphenyl)phenyl]piperidine-2-carboxamide
4-({1-[(3-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
N-methyl-N-(1-methylpiperidin-4-yl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
(2S)-2-{[4-methyl-7-(methylsulfanyl)quinolin-2-yl]amino}propan-1-ol
2-oxo-6-(propan-2-yl)-N-[1-(thian-4-yl)piperidin-4-yl]-1,2-dihydropyridine-3-carboxamide
methyl 5-{[(3,4-difluorophenyl)methyl]amino}-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(furan-2-ylmethyl)-2-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}acetamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
methyl[2-(morpholin-4-yl)ethyl](2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
5-{3-[5-(4-methylphenyl)furan-2-yl]propanoyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-3-(methanesulfonylmethyl)piperidine
2-(3-fluorophenyl)-N-({7-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]thiophene-2-carboxamide
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(5-methylthiophen-2-yl)methyl]amine
[3-(hydroxymethyl)-4-[3-(morpholin-4-ylmethyl)phenyl]phenyl]methanol
5-[3-(3-methylphenoxy)azetidine-1-carbonyl]quinoxaline
1-(2-methyloxolane-2-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(4-{[3-(1,2-oxazinane-2-carbonyl)-1,2-oxazol-5-yl]methoxy}phenyl)ethan-1-one
dimethyl({1-[(1-pentylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)amine
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(thiophen-2-yl)butanamide
1-(2-amino-5-ethylpyrimidin-4-yl)-4-(pyridin-3-yl)piperidin-4-ol
N-(1-methoxypropan-2-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
5-cyclopropanecarbonyl-1'-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-cyclopentyl-1-[1-(3-phenylpropyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide