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5-(2-fluorophenoxymethyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
3-(2-methyl-1H-indol-1-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
1-{4-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-2-(methylamino)ethan-1-one
{4-[3-(dimethylamino)benzoyl]-1,4-oxazepan-6-yl}methanol
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
ethyl 3-(2-methoxyethyl)-1-(oxan-4-yl)piperidine-3-carboxylate
(1R,5S,6R)-3-(quinolin-4-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
2-[(4,8-dimethyl-2-oxo-2H-chromen-7-yl)oxy]-N-[(1-methylpyrrolidin-3-yl)methyl]acetamide
1-{1-[2-(4-chlorophenyl)acetyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
4-[4-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
(3S,4S)-1-(benzenesulfonyl)-4-[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]pyrrolidin-3-ol
4-{2-[2-(pyridin-2-yl)piperidine-1-carbonyl]phenyl}morpholine
1-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]-1,2,3,4-tetrahydroquinolin-2-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2,2,2-trifluoroethyl)-1,3-oxazole-4-carboxamide
2-{[(1,4-dithiepan-6-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-methyl-4-(3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}phenyl)butan-2-ol
[(3R,4R)-4-(azepan-1-ylmethyl)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}pyrrolidin-3-yl]methanol
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-[3-(4-hydroxyphenyl)propyl]urea
1-[(diethylcarbamoyl)methyl]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-5-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
10-[4-(pyridin-3-yl)piperazine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
N4-[2-(3,5-dimethylphenoxy)ethyl]-N4,5-dimethylpyrimidine-2,4-diamine
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl](2-methylpropyl)(thiophen-3-ylmethyl)amine
6-[4-(6-ethylpyrimidin-4-yl)piperazine-1-carbonyl]-1-methyl-1H-indole
2-[9-(2-fluoro-4-methylbenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
4-(2,4-dioxoimidazolidin-1-yl)-N-(2-methylpropyl)-N-(pyridin-4-ylmethyl)benzamide
5-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
4-[2-(azocan-1-yl)acetyl]-1-(4-methylphenyl)piperazin-2-one
3-(2-ethyl-1H-imidazol-1-yl)-1-[2-(4-fluorophenyl)morpholin-4-yl]propan-1-one
methyl 3-({4-[2-(methylsulfanyl)benzoyl]-7-oxo-1,4-diazepan-1-yl}methyl)benzoate
3-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
1-cyclopentyl-N-[(3-methoxyphenyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
(1-methyl-1H-imidazol-2-yl)({1-[(2,6,8-trimethylquinolin-4-yl)methyl]piperidin-4-yl})methanol
3-{2-[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
4-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-oxazepane
5-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
4-{[5-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-1-yl]methyl}pyridine
3-(2,3-dihydro-1H-isoindol-2-yl)-N-[(1-methylpyrrolidin-3-yl)methyl]benzamide
2-(2-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
3-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]thiophene-2-carboxamide
2-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
3-(3-chloro-5-fluorophenyl)-1-[(4-methyl-1,4-oxazepan-6-yl)methyl]urea
N-[2-chloro-5-(diethylcarbamoyl)phenyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-(piperidin-1-yl)pyrimidine
4-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-fluoropyridine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-[3-(cyclohexyloxy)propyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-(2-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
N-[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]benzamide