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3-methyl-1-propyl-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-4-carboxamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
4-[6-(1-hydroxyethyl)pyridin-2-yl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(4-carbamoylpiperidin-1-yl)-2-[4-(methylsulfanyl)phenyl]acetic acid
6-(4-chlorophenyl)-N-(oxan-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-(2-hydroxyphenyl)ethan-1-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
4-{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}-3-methylpiperazin-2-one
7-(cyclopropylmethyl)-2-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2,3-thiadiazole-5-carboxamide
2-ethyl-8-[4-(4-methoxyphenyl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
ethyl 4-{2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetyl}piperazine-1-carboxylate
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
3-[(2,4-dimethoxyphenyl)methyl]-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl]sulfamoyl})amine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1,2-oxazole-3-carboxamide
4-{[3-(5-chloro-2-methoxybenzoyl)piperidin-1-yl]methyl}pyridine
(3R)-1-({1-[1-(quinolin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-3-ol
1-(3-acetylphenyl)-3-(1-cycloheptylpiperidin-3-yl)urea
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}acetamide
6-methyl-5-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}quinoline
2-{1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]pyrrolidin-2-yl}-1,3-thiazole
1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-4-phenylpiperidine-4-carbonitrile
methyl 3-(7-chloro-2-{[3-(1H-1,2,4-triazol-1-yl)propanamido]methyl}-2,3-dihydro-1-benzofuran-5-yl)benzoate
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-propylpiperidin-4-yl)acetamide
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
3-({methyl[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)benzonitrile
5-(2-methoxyphenoxymethyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
(2E)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-3-phenylprop-2-en-1-one
N-(oxolan-2-ylmethyl)-1-phenyl-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
N,2,4-trimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-thiazole-5-carboxamide
6-[3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
(1R,3S)-3-(2-hydroxyethoxy)-7-(3-methyl-1H-pyrazole-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
1-(oxolane-2-carbonyl)-4-(5-phenyl-1,2-oxazole-3-carbonyl)piperazine
(5S,9aS,9bS)-5-(6-chloro-2H-chromen-3-yl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-indol-3-yl)propanamide
3-cyclopropyl-1-(3,4-dimethylphenyl)-5-[1-(ethanesulfonyl)ethyl]-1H-1,2,4-triazole
(2S,4S)-4-amino-N-ethyl-1-(2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}acetyl)pyrrolidine-2-carboxamide
2-cyclopropyl-8-(6-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-N-(3-methylphenyl)propanamide
1-(1-methyl-1H-pyrazole-3-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-6-methyl-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-phenyl-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-1H-1,2,3-triazole
N-[2-(2-chloro-4-methylphenoxy)ethyl]-1-(2-methoxyethyl)-N-methylpyrrolidine-3-carboxamide
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-[(2-methylphenyl)sulfanyl]ethan-1-one