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1-methanesulfonyl-4-[3-(1H-pyrazol-4-yl)benzoyl]-1,4-diazepane
1-cyclobutanecarbonyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]piperidine-4-carboxamide
1-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
2-[2-({[(3-methoxyphenyl)methyl](methyl)amino}methyl)phenyl]-5,6-dimethyl-3,4-dihydropyrimidin-4-one
(2R,6S)-4-[2-(4-chlorophenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-2,6-dimethylmorpholine
2-methyl-N-[3-(pyridin-3-yloxy)propyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
4-(4-fluorophenyl)-1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,2,3,6-tetrahydropyridine
4-(4-fluorophenyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-4-oxobutanamide
N-methyl-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(oxan-4-yl)pyridin-2-amine
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}pyrrolidin-2-one
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-cyclopropyl-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(2-phenylethyl)-N-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
7-[(4-fluorophenyl)methyl]-6-oxo-N-(prop-2-en-1-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-4,4-difluoropiperidine
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]urea
5-{[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-(3-methyl-1,2-oxazole-5-carbonyl)-8-azabicyclo[3.2.1]octane
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-pyrazol-1-yl)benzamide
1-[(3-fluorophenyl)methyl]-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-2-one
1-benzyl-4-[2-(ethylsulfanyl)pyrimidin-5-yl]-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[2-(morpholin-4-yl)ethyl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
4-(1H-1,3-benzodiazol-2-yl)-1-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(azocan-1-yl)-3-[2-methoxy-4-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
ethyl 4-[1-(1-methyl-1,2,3,4-tetrahydroquinoline-6-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
{1-[({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]cyclobutyl}methanol
4-benzyl-1-[(6-methylpyridin-2-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4R)-4-{[(3-methoxyphenyl)methyl]amino}-N-methyl-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
[(6-chloropyridin-3-yl)methyl][(3-methoxyphenyl)methyl](prop-2-en-1-yl)amine
4-[(1-benzylpyrrolidin-3-yl)amino]-N-ethylpiperidine-1-carboxamide
N-ethyl-3-methyl-4-[({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}carbamoyl)amino]benzamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-(3-methoxyphenyl)-N-methyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]({[2-(2-methoxyethyl)pyrimidin-5-yl]methyl})methylamine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}isoquinoline-5-carboxamide
N-cyclopropyl-1-{2-[(3-methoxyphenyl)sulfanyl]acetyl}piperazine-2-carboxamide
(3S,4S)-4-(propan-2-yloxy)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-ol
N-[1-(4-methoxyphenyl)ethyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
2-(2,2-dimethyloxan-4-yl)-1-(2-phenylethyl)-1H-imidazole
[(4-tert-butylphenyl)methyl](1H-imidazol-2-ylmethyl)methylamine
N-(adamantan-1-ylmethyl)-N-methyl-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
5-[1-(furan-3-ylmethyl)-4-hydroxypiperidin-4-yl]-N-(2-methoxyphenyl)-1-benzofuran-2-carboxamide
N-{4-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-4-oxobutyl}acetamide