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(1R,9S)-5-amino-3-(3-fluoro-4-methoxyphenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
(1R,7S)-3-(2-ethylbutyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(4aR,8aS)-1-(2,6-dimethylquinoline-4-carbonyl)-6-(4-fluorobenzoyl)-decahydro-1,6-naphthyridine
[(3R,4S)-1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-3-(2-methoxyphenyl)propanamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)oxane-4-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[3-(methylsulfanyl)propyl]-2,7-diazaspiro[4.5]decan-6-one
3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]-1-[3-(1H-pyrazol-1-yl)phenyl]urea
1-[(3,5-dimethylphenyl)methyl]-4-[2-(methylsulfanyl)propanoyl]piperazin-2-one
2-methyl-2-{2-[(1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}propanoic acid
1-methyl-4-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetyl}piperazine-2-carboxylic acid
1-(2-methoxyethyl)-3,8-bis[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3,4,5-trifluorophenyl)methyl]-1,4-dioxane-2-carboxamide
methyl (2S)-1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidine-2-carboxylate
methyl 3-[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)carbamoyl]benzoate
1-[(2,3-difluorophenyl)methyl]-4-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}piperidine
1-[2-methoxy-4-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
5-{[methyl(oxan-2-ylmethyl)amino]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
2-[4-(propane-1-sulfonyl)morpholin-3-yl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
5-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}benzenesulfonamide
methyl 3-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}propanoate
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-({[(3-methylphenyl)methyl]amino}methyl)piperidin-2-one
5-[1-methyl-5-(piperidin-1-yl)-1H-1,2,4-triazol-3-yl]-1H-indole
3-[(benzylamino)methyl]-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
methyl(2-phenylethyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
3-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-3-(1H-pyrazol-5-yl)piperidine
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(quinolin-6-ylmethyl)amine
1-(4-cyano-2-fluorophenyl)-3-[3-(2-ethyl-1H-imidazol-1-yl)propyl]urea
2-(4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
1,4-dimethyl 2-({6-phenylimidazo[2,1-b][1,3]thiazol-3-yl}formamido)butanedioate
1-(2-cyclohexylethyl)-N-ethyl-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
methyl({1-[4-(quinolin-5-yl)phenyl]propyl})amine
5-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
1-{3-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
3-[2-({3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)ethyl]-1,3-oxazolidin-2-one
N-(2-methoxyethyl)-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-4-carboxylate
3-({[3-(1H-indazol-1-yl)propyl]amino}methyl)pyrrolidin-3-ol
4-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-3-yl]-5-phenyl-2-(pyridin-4-yl)pyrimidine
5-(1H-imidazol-1-ylmethyl)-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)ethan-1-one
2-[(3-fluorophenyl)methyl]-4-{4-[2-(4-phenylphenyl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amine
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-N'-[2-(methylsulfanyl)phenyl]butanediamide
2-[3-oxo-9-(oxolan-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetamide