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1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyphenoxy)piperidine
N-{1-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
methyl 4-(5-{[(3-hydroxy-3-methylbutyl)(methyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
2-({[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)amino)-1-phenylethan-1-ol
N-butyl-N-methyl-3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
2-[(3,4-dihydro-2H-1-benzopyran-2-ylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(1S,5R)-3-cyclobutanecarbonyl-6-(2-fluorobenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(3-fluoro-2,4-dimethylphenyl)methyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
6-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-1-methyl-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-4-one
1-benzyl-N5-cyclopropyl-N3-methyl-4-oxo-N3-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(4-fluorophenyl)-N-[2-(furan-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[(5-propylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
5-{[(2S)-2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-2-(2-methylphenyl)pyrimidine
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
1-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
N-methyl-N-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}aniline
3-benzoyl-1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidine
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2-ethylbutanamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(pent-4-enoyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[(3-{2-[4-(2H-1,3-benzodioxole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]morpholine
3-(2-fluorophenyl)-3-{[3-(2-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}propanoic acid
4-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-{8-cyclopentyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-methoxypyridine-3-carbonitrile
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(methyl)({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amine
1-{1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}-2-phenylethan-1-one
7-(1,3-benzothiazol-2-yl)-4-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2,2-dimethylbutan-1-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-(3-phenylprop-2-yn-1-yl)-N-propylacetamide
N-[2-(4-{[2-(2H-1,2,3-benzotriazol-2-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]cyclobutanecarboxamide
2-(3-phenylpiperidin-1-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
4-(2-aminoacetyl)-5-benzyl-1-(3-phenylphenyl)piperazin-2-one
N-[(3S,4R)-1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-4-propylpyrrolidin-3-yl]acetamide
N-[4-(1H-1,2,3,4-tetrazol-5-yloxy)phenyl]thian-4-amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-5-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(3-chloro-4-methoxyphenyl)-6-(2-ethylbutyl)-6-azaspiro[2.5]octane-1-carboxamide
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}cyclopropanecarboxamide
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butan-1-one
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-(1,3-thiazol-2-ylmethyl)piperidine
5-ethyl-1'-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(methylamino)-N-propyl-N-(pyridin-3-ylmethyl)benzamide
3-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
(3S,4R)-3-benzyl-1-(5,6-dimethylpyrimidin-4-yl)-4-methylpiperidin-4-ol
(3R)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3,4,4-trimethylpyrrolidin-3-ol
5-chloro-3-methyl-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
4-methyl-6-{4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}pyrimidin-2-amine
1-[1-(5-chloropyridine-2-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
7,8-dimethyl-4-(4-methylpiperidine-1-carbonyl)-2-(2-methylpyrimidin-5-yl)quinoline
(2R)-N1-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]pyrrolidine-1,2-dicarboxamide