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N-[(5-methylpyrazin-2-yl)methyl]-2-(1-propylpiperidin-4-yl)acetamide
N-(3-hydroxy-3-phenylpropyl)-N,2,6-trimethylpyridine-4-carboxamide
1-[2-(pyridin-2-yl)pyrrolidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
5-(2-fluorophenoxymethyl)-N-[1-(furan-2-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
(3S,4S)-1-[(1,5-dimethyl-1H-indol-2-yl)methyl]-4-(dimethylamino)pyrrolidin-3-ol
1-cyclopentyl-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]piperidine-3-carboxamide
3-(1H-imidazol-2-yl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]benzamide
2-amino-4-(5-cyano-1-ethyl-1H-pyrrol-3-yl)-6-(4-hydroxy-3-methoxyphenyl)pyridine-3-carbonitrile
4-ethyl-3-{1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
4-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine
(4aR,8aS)-6-[(3-ethoxy-4-methoxyphenyl)methyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
N-(oxolan-2-ylmethyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}propanamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-4H-thieno[3,2-b]pyrrole-5-carboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
5,8-dichloro-3-[2-(4-hydroxy-1-methylpiperidin-4-yl)ethyl]-3,4-dihydroquinazolin-4-one
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
2-({4-[3-(2,5-dioxoimidazolidin-4-yl)propanoyl]piperazin-1-yl}methyl)benzonitrile
2-methyl-6-[5-(oxolan-3-ylmethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]-1,3-benzothiazole
3-fluoro-N-[2-(furan-2-ylmethoxy)phenyl]-4-methoxybenzamide
6-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-3-ethyl-3H-imidazo[4,5-b]pyridin-2-amine
1-(6-aminopyrimidin-4-yl)-4-(oxane-4-carbonyl)-1,4-diazepan-6-ol
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-2-methoxy-N-(oxolan-2-ylmethyl)benzamide
2-[4-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]phenol
2-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-6-methylquinolin-4-ol
ethyl 1-[cyclopropyl(3-methylpyridin-2-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
4-{[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-1H-indole
3-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1-{[1-(2-phenylethyl)piperidin-4-yl]methyl}urea
1-(furan-2-ylmethyl)-4-[3-(3-methylphenoxy)azetidine-1-carbonyl]piperidine
(4aR,8aR)-2-cyclopentanecarbonyl-7-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-decahydro-2,7-naphthyridin-4a-ol
1-cyclopropyl-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-pyrrole-2-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethylacetamide
2-amino-4-(1-methyl-3-phenyl-1H-pyrazol-4-yl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{3-[3-(pyridin-4-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
2-tert-butyl-6-(4-chloro-2-methylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-[(4aR,8aR)-4a-hydroxy-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-2-yl]-2-phenylethan-1-one
1-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-(5-{[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1H-imidazole-2-carboxamide
3-cyclopentyl-5-(1-ethylpiperidin-4-yl)-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
5-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-2-ethylpyrimidine
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-2-(morpholine-4-carbonyl)pyridin-4-amine
ethyl 3-[(2-methylphenyl)methyl]-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine-3-carboxylate
1-{4-[({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]phenyl}pyrrolidin-2-one
(3R,4R)-3-cyclobutyl-4-methyl-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)pyrrolidin-3-ol
2-(2-{1-[(3-phenyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide