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3-(2-{[1-(3-phenylphenyl)piperidin-4-yl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(2-chlorophenyl)ethan-1-one
1-(3,5-dimethyl-1H-pyrazole-4-carbonyl)-3-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(propan-2-yl)pyridine-4-carboxamide
3-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
2-({[(3R,4R)-4-(hydroxymethyl)-1-(4-methyl-1,3-oxazole-5-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-methyl-6-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
7-(5-methylthiophen-2-yl)-4-[3-(pyridin-3-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
1-{2-[(4aS,8aR)-2-oxo-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}-1-methylurea
2-{[2-(furan-2-yl)pyrrolidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-[3-(3-methylphenyl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
(2S,4R)-N-ethyl-1-(1-propylpiperidin-4-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-methyl-4-{[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-N-propyl-1,4-dihydroquinoline-3-carboxamide
ethyl({[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-methoxy-1-[1'-(6-methylpyridazin-3-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-(4-methylphenoxy)piperidine-4-carboxylic acid
7-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-(methylsulfanyl)pyrimidine
N-{4-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]phenyl}acetamide
methyl 8-(2-methylpropyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[1-(4-chlorobenzoyl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(2-fluorophenyl)methyl]propanamide
1-ethyl-3-(2-methylpropyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
1-(diethylamino)-3-[2-methoxy-4-({[(4-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N3-methyl-N5-[(4-methylphenyl)methyl]-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-[(2-chlorophenyl)methyl]-N,N-bis(prop-2-en-1-yl)-1,2-oxazole-5-carboxamide
(1S,5R)-3-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4S)-4-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-1-(1,4-dithiepan-6-yl)pyrrolidin-3-ol
(2S,4S,5R)-4-[(2-acetamidoethyl)carbamoyl]-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
(3aR,5R,6S,7aS)-2-[1-(pyridine-2-carbonyl)piperidin-4-yl]-octahydro-1H-isoindole-5,6-diol
2-{4-[(2-ethylpyrimidin-4-yl)methyl]piperazin-1-yl}-1,3-benzoxazole
2-(5-{1-[(1-methylpyrrolidin-3-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)benzonitrile
(1S)-1-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pentane-1,5-diamine
4-(3,4-dimethylphenyl)-3-(piperidin-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
1-({[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)cyclohexan-1-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methylbenzamide
1-[4-({[3-(dimethylamino)propyl]amino}methyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
6-(2-chlorophenyl)-7-methyl-8-oxo-N-(pentan-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2,7,8-trimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]quinoline-4-carboxamide
2-amino-N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-4-ethyl-1,3-thiazole-5-carboxamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]acetamide
1-(cyclohexylmethyl)-4-(4-methanesulfonylphenyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-({3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)-2-(piperidin-1-yl)pyrimidine
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-4-(morpholin-4-yl)butan-1-one
7-[2-(2-fluorophenyl)acetamido]-N-(prop-2-en-1-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide