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2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
1-(1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[3-(1H-1,2,3-triazol-1-yl)propyl]propanamide
[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1H-indole-6-carbonyl)piperidin-3-ol
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-ethylpiperidine-4-carboxamide
(1S,5R)-3-[(3-fluoro-4-methoxyphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(cyclohexylmethyl)-N5-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
[(3R,4R)-1-(3-chloro-4-methylbenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-[(3-hydroxyphenyl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
1-(2-cyclohexylethyl)-3-hydroxy-3-({[2-(2-oxoimidazolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
methyl 3-[(2,6-difluorophenyl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-methyl-4-(4-methylpyrimidine-5-carbonyl)-3-(propan-2-yl)piperazin-2-one
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(2,2,2-trifluoroethyl)piperazin-1-yl]ethan-1-one
5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-(propan-2-yl)piperidine-4-carboxamide
ethyl 4-[(4-{[1-(4-fluorophenyl)ethyl]amino}quinazolin-2-yl)methyl]piperazine-1-carboxylate
(2S,4S)-4-{2-[(dimethylcarbamoyl)amino]acetamido}-N-ethyl-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
7,7-dimethyl-2-[1-(pyrrolidin-1-ylmethyl)cyclopropyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(4-chlorophenyl)-N-[(4-methanesulfonylmorpholin-2-yl)methyl]butanamide
1-(1H-indol-5-ylmethyl)-4-(oxan-4-yl)-1,4-diazepan-6-ol
N-[(4-fluorophenyl)methyl]-1-methyl-N-(1-phenylethyl)-1H-imidazole-5-carboxamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-5-propylthiophene-3-carboxamide
N-[3-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]cyclopropanecarboxamide
1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(3aS,7aR)-2-(1-benzofuran-5-ylmethyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
(2S,4R)-1-(naphthalen-1-ylmethyl)-N-(propan-2-yl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-amino-4-(2,3-dimethoxyphenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
3-[4-(1-methylpiperidin-4-yl)piperidine-1-carbonyl]pyridazine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
3-methyl-1-propyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1H-pyrazole-4-carboxamide
3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-6-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-amino-N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-6-methylpyrimidine-4-carboxamide
8-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(1R,3S)-3-{[2-(1-benzylpiperidin-4-yl)ethyl]carbamoyl}cyclopentane-1-carboxylic acid
3-{1-[1-(pyridin-2-yl)piperidine-3-carbonyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-(propan-2-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-4-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
3-(1H-1,3-benzodiazol-1-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]propanamide
2-[(3-ethoxypropanamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
8-methyl-3-[2-(4-phenylpiperidin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
4-[(benzyloxy)methyl]-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-{2-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-indole
3-(2-amino-1,3-thiazol-4-yl)-1-{spiro[indene-1,4'-piperidine]-1'-yl}propan-1-one
2-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
N-[1-(pentan-2-yl)-1H-pyrazol-5-yl]-2-(2-propyl-1H-imidazol-1-yl)acetamide
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
4-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-phenylpiperazin-2-one