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N3-methyl-4-oxo-1-(3-phenylpropyl)-N5-{[4-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
2-(2,3-dimethoxyphenyl)-5-methyl-4-{[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-oxazole
3-(3-methoxyphenyl)-5-{[1,2,4]triazolo[1,5-a]pyrimidin-6-ylmethyl}-1,2,4-oxadiazole
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-5-oxopyrrolidine-2-carboxamide
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclopentyl-5-oxo-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]pyrrolidine-3-carboxamide
1-ethyl-N,N-dimethyl-3-{4-[1-(piperidin-1-yl)ethyl]phenyl}-1H-1,2,4-triazol-5-amine
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-2-(4-fluorophenyl)-N-(2-methoxyethyl)acetamide
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
2,4-difluoro-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)benzamide
3-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]benzonitrile
5-(2-methylpropyl)-1'-(1,3-thiazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{methyl[(1-methylpyrrolidin-2-yl)methyl]amino}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-(2H-indazol-2-yl)ethan-1-one
6-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-N,N-dimethylpyrazine-2-carboxamide
3-(dimethylamino)-N-(3-fluoro-5-methylphenyl)pyrrolidine-1-carboxamide
6-ethyl-1,5-dimethyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(furan-2-carbonyl)-4-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}-1,4-diazepane
N-benzyl-3-[(thiophen-2-ylformamido)methyl]piperidine-1-carboxamide
2-{[2-methyl-2-(morpholin-4-yl)propyl]amino}pyridine-3-carbonitrile
4-methoxy-6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidin-2-amine
2-[methyl({4-methyl-5-[1-(pyridine-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-3-azaspiro[5.5]undecan-9-amine
N-({7-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-fluorobenzamide
8-(1-benzyl-1H-pyrazole-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(thiophene-2-sulfonamido)acetamide
4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1-[(3-methylphenyl)methyl]piperazin-2-one
5-(5-chloro-2-methoxyphenyl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
3-phenyl-1-[1-(2-phenylacetyl)piperidin-3-yl]propan-1-one
5-(4-methylphenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]pent-4-enamide
(4aS,7aR)-1-(4-ethylbenzoyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-4-amino-N-[(4-chlorophenyl)methyl]-N-(3-hydroxypropyl)-1-methylpyrrolidine-2-carboxamide
(2S,4R)-4-hydroxy-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(4-methylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-{1-[1-(2-amino-2-methylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
4-[(2,3-dimethoxyphenyl)methyl]-3-[2-oxo-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]piperazin-2-one
methyl 6-(2-cyclopentylacetyl)-2-[(4-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[2-({dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)ethyl]-1,2,3,4-tetrahydrophthalazine-1,4-dione
9-{2-[4-(hydroxymethyl)phenyl]acetyl}-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(4aR,8aR)-2-cyclobutanecarbonyl-7-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-decahydro-2,7-naphthyridin-4a-ol
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-5-(oxolan-2-yl)thiophene-2-carboxamide
4-[(dimethylamino)methyl]-1-[4-(3-fluorophenyl)benzoyl]azepan-4-ol
5-(4-ethylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-[1-(3-methylpyridin-2-yl)-1H-pyrazol-4-yl]ethan-1-ol
4-(2-ethylpyrimidine-5-carbonyl)-1-(4-methoxyphenyl)piperazin-2-one
2-amino-4-(2-ethylpyrimidin-5-yl)-6-phenylpyridine-3-carbonitrile
4-[3-cyclopropyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1-oxaspiro[4.4]nonan-2-one