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2-{9-oxa-2-azaspiro[5.5]undecan-2-ylmethyl}benzonitrile
N-(2-ethoxyphenyl)-N'-methyl-N'-[1-(pyridin-3-yl)propyl]propanediamide
1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
methyl 2-(2-amino-6-methylpyrimidin-4-yl)benzoate
N-({5-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
2-[5-(2,3-dimethylquinoxaline-6-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
5-[3-(3-methoxypropyl)piperidine-1-carbonyl]-2-(trifluoromethyl)-1H-1,3-benzodiazole
8-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-5-(ethoxymethyl)quinoline
ethyl 5-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
(3S,4R)-4-(hydroxymethyl)-1-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}piperidin-3-ol
3-(3-methoxy-4-methylphenyl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
9-[(5-chloro-2-fluorophenyl)methyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-1-{3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
5-{[methyl({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}pyrimidin-2-amine
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-methoxybenzamide
6-methyl-2-phenyl-N-[1-(pyridin-2-yl)propan-2-yl]pyrimidin-4-amine
N-cyclopropyl-5-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(thiophen-2-yl)acetamide
2-{1,4-bis[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}ethan-1-one
3-({4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}methyl)benzoic acid
2-({2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-oxoethyl}sulfanyl)-6-methyl-3,4-dihydropyrimidin-4-one
(1R,5R)-6-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4R)-1-[(5-carboxyfuran-2-yl)methyl]-4-(2,3-dimethoxyphenyl)pyrrolidine-3-carboxylic acid
N-{2-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}acetamide
methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl}){[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
N-[1-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2-methylbenzamide
1-{4-[(2-phenylpropyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-[4-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]-1,3-benzothiazole
(butan-2-yl)(3-phenylprop-2-yn-1-yl)(1,3-thiazol-2-ylmethyl)amine
N-[1-benzyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-1,2-oxazole-3-carboxamide
7-(cyclobutylmethyl)-2-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(dimethylamino)-2-methylpropyl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
3-{[(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)oxy]methyl}pyridine
2-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}(thiophen-2-ylmethyl)amino)butan-1-ol
4-tert-butyl-2-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)phenol
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(pyridin-4-yl)propanamide
7-(1,3-benzothiazol-2-yl)-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-(4-chlorophenyl)-N-methyl-N-(3-methylbutyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
4-{3-[(4-fluorophenyl)amino]piperidine-1-carbonyl}-N,N-dimethylpiperidine-1-carboxamide
3-propyl-4-[2-(propylsulfanyl)pyrimidin-5-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-amino-1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
2-(3-hydroxyphenyl)-1-(3-propoxypiperidin-1-yl)ethan-1-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
1-(2-fluorophenyl)-4-{1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}piperazine
N-[(3-methyloxetan-3-yl)methyl]-3-phenoxypropanamide