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2-(2-{1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-(1,4-dithiepan-6-yl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
2-methyl-4-(4-{[3-(piperidin-1-ylmethyl)piperidin-1-yl]methyl}phenyl)butan-2-ol
1-(1-methylpiperidin-4-yl)-4-{[2-(trifluoromethoxy)phenyl]methyl}piperazine
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
2-methyl-1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine
4-chloro-1,5-dimethyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1H-pyrazole-3-carboxamide
1-[4-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)thiophen-2-yl]ethan-1-one
N-[(4-fluorophenyl)methyl]-9-hydroxy-N-(1-methoxypropan-2-yl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
8-chloro-2-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)quinolin-4-ol
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
2-oxo-1-phenyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxamide
(1-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-3-yl)methanol
5-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2-(propan-2-yl)-1,3-benzoxazole
6-(3-acetamidopyrrolidin-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
(3aR,6aR)-2-cyclopentyl-N-[2-(pyridin-3-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-(1-ethylpiperidin-4-yl)-2,7-diazaspiro[4.5]decane
4-{[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperidin-4-yl]oxy}pyridine
3-methyl-2-oxo-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2,3-dihydro-1,3-benzoxazole-6-sulfonamide
7-chloro-4-[3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3,3-dimethylbutan-1-one
(2S,4S)-4-amino-N-ethyl-1-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)pyrrolidine-2-carboxamide
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
N-cyclopentyl-7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
1-cyclopentyl-N-methyl-5-oxo-N-(quinoxalin-2-ylmethyl)pyrrolidine-3-carboxamide
7-(2-methoxyethyl)-2-{[4-(methylsulfanyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
N-methyl-2-(2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamido)acetamide
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]ethan-1-one
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-cyclohexyl-1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)-N-methylpiperidine-4-carboxamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-methyl-5-{1-[3-(6-methylpyridin-2-yl)propyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazole
(2S)-2-[1-(2,4-difluorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]pyrrolidine-1-carboxamide
N-{[1-(3-cyanopyridin-2-yl)piperidin-3-yl]methyl}-2-(4-methoxyphenyl)acetamide
methyl(2-phenylethyl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(2S)-2-amino-4-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]butanoic acid
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
1-[(3-ethoxy-4-hydroxyphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-methyl-7-oxo-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
2-{[benzyl(methyl)amino]methyl}-4-(pyrimidin-2-yl)phenol
2-hydroxy-3-methoxy-N-[2-(pyridin-3-yloxy)propyl]benzamide
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-[(oxan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-3-yl]acetamide
N-(dicyclopropylmethyl)-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
3-chloro-N,6-dimethyl-N-[3-(3-methylphenoxy)propyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
6-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-4-amine
4-(4-chlorophenyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]butanamide
2-[4-(5-methoxypyridin-3-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide