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1-(2-methylphenyl)-4-[1-(pyridine-2-carbonyl)piperidin-3-yl]piperazine
1-phenyl-2-({8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}amino)ethan-1-ol
1-(cyclohexylmethyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
2-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1,3-benzothiazole-5-carboxamide
3-[3-({[1-(carbamoylmethyl)piperidin-4-yl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
N-methyl-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]-N-(quinolin-8-ylmethyl)acetamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidine-3-carboxylate
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(quinoxalin-2-yl)-decahydro-1,6-naphthyridin-2-one
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrrole
ethyl 4-[(3-fluorophenyl)methyl]-1-(5-methylpyrazine-2-carbonyl)piperidine-4-carboxylate
N-[2-(azepane-1-carbonyl)phenyl]-2-hydroxypyridine-3-carboxamide
(3S,4R)-4-(3-methoxyphenyl)-1-(oxan-4-ylmethyl)pyrrolidine-3-carboxylic acid
3-{1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine-3-carbonyl}pyridine
1-(oxane-2-carbonyl)-4-phenylpiperidine-4-carbonitrile
3,5-dimethyl-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]adamantane-1-carboxamide
methyl 3-(2H-1,3-benzodioxole-5-carbonyl)-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(4-acetyl-1,4-diazepan-1-yl)-3-(3-chlorophenyl)-3-phenylpropan-1-one
N-methyl-2-{methyl[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}propanamide
3-(4-fluorophenyl)-4-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}-1H-pyrazole
1-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]-3-methylimidazolidin-2-one
2-(3-hydroxypropyl)-8-[(5-methylthiophen-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-ethyl-N-[(4-methylphenyl)(pyridin-4-yl)methyl]pyrimidine-5-carboxamide
3-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanoic acid
3-amino-1-{[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]methyl}pyrrolidine-3-carboxylic acid
4-methyl-5-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]-N-[(2,3,4-trimethoxyphenyl)methyl]-1,3-thiazol-2-amine
methyl 6-[(3,5-dimethylphenyl)methyl]-2-[(propan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{3-[(3S,4R)-3-acetamido-4-(4-methylphenyl)pyrrolidin-1-yl]propoxy}benzamide
1-{3-[(3-methoxypiperidin-1-yl)sulfonyl]benzoyl}-4-methylpiperazine
(2S,4R)-4-amino-N-ethyl-1-[3-(furan-2-yl)propanoyl]pyrrolidine-2-carboxamide
9-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2,3,6-trimethyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]quinoline-4-carboxamide
14-[3-(pyridin-2-ylmethoxy)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-(4-methylpyridin-3-yl)-2-{4-[(2-phenyl-1,3-oxazol-4-yl)methyl]morpholin-3-yl}acetamide
[(3R,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methanol
3-(1H-pyrazol-1-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
N-(2-methoxyethyl)-3-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}propanamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
4-[2-(5-acetylthiophen-3-yl)acetyl]-3-(3-fluorophenyl)piperazin-2-one
2-{1-[(2,4-dimethoxy-3-methylphenyl)methyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
N-(2-methylpropyl)-1-{1-[(2,3,4-trimethoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
1-[4-(piperidin-3-yl)benzoyl]-4-(pyrimidin-2-yl)-1,4-diazepane
6-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole
N-[5-(2-ethoxyethyl)-1,3,4-thiadiazol-2-yl]-4-phenylazepane-1-carboxamide
8-chloro-2-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)quinoline
5-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-cyclohexyl-4-[2-(2-methoxyethyl)-1,3-benzoxazole-6-carbonyl]piperazin-2-one
1-(4-chlorophenyl)-3-[1-(morpholine-4-carbonyl)piperidin-4-yl]urea
4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1-ethyl-3-methylpiperazin-2-one
1-(4-chlorophenyl)-3-methyl-3-[2-(oxan-4-yl)ethyl]urea
2-(ethylsulfanyl)-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide