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2-methoxy-N-{2-methyl-3-[({[1-(pyrrolidin-1-yl)cyclopentyl]methyl}carbamoyl)amino]phenyl}acetamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(propane-2-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
1-cyclohexanecarbonyl-2-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}pyrrolidine
1-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1,2-dihydroquinoxalin-2-one
N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2S)-2-acetamido-3-(1H-imidazol-4-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)propanamide
1-[3-(3-{[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]methyl}phenoxy)-2-hydroxypropyl]piperidin-4-ol
N-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
[(4-{2-[2-(dimethylamino)ethoxy]phenyl}phenyl)methyl]dimethylamine
(1S,9S)-11-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-(2-methoxyethyl)-6-oxo-N-{[2-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2-{4-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]phenyl}-2-methylpropanamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]amino}methyl)piperidin-2-one
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
(3S)-1-(1,3-benzothiazol-2-yl)-N,N-dimethylazepan-3-amine
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-2,4-dimethylpyrimidine
4-[(3,5-difluorophenyl)methyl]-1-phenylpiperazin-2-one
2-ethoxy-5-[2-(4-methylpiperazin-1-yl)pyrimidin-4-yl]benzoic acid
N-(4-chloro-3-fluorophenyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carboxamide
N-methyl-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}-N-(quinoxalin-6-ylmethyl)benzamide
4-tert-butyl-N-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]benzene-1-sulfonamide
1-benzyl-8-[3-(5-methylfuran-2-yl)butyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 2-(5-methyl-2-{[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)formamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
1-ethyl-N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-{6-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]pyridin-3-yl}ethan-1-one
2-(2,1,3-benzoxadiazole-4-sulfonyl)-8-methyl-2,8-diazaspiro[4.5]decane
3-(1-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carbonyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
3-ethoxy-1-[3-(3-methylphenoxy)azetidin-1-yl]propan-1-one
[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
1-cyclopropyl-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-5-oxopyrrolidine-3-carboxamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]acetamide
N-(2,4-dimethoxyphenyl)-3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-1,2,4-triazole-5-carboxamide
4-{6-[3-(pyridin-4-yl)azetidin-1-yl]pyrimidin-4-yl}morpholine
1-(1H-indol-2-ylmethyl)-4-(pyridin-4-yl)-1,4-diazepan-6-ol
2-[benzyl({[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
N-methyl-3-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl][1-(2-methyl-1H-imidazol-1-yl)propan-2-yl]amine
1-{4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
2-{4-[(2-methoxyethyl)(methyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}pyridine-3-carbonitrile
{1-[(2-methoxyphenyl)methyl]-3-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
N-(3,4-dimethoxyphenyl)-1-[(2,5-dimethoxyphenyl)methyl]piperidin-3-amine
2-(2-phenyl-1,3-thiazol-4-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
N-cyclopropyl-N-[(4-methoxyphenyl)methyl]-5-methylthiophene-2-carboxamide
2-cyclopropyl-5-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]pyrimidin-4-ol
3-(3-methylthiophene-2-carbonyl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
3-cyclobutyl-4-(2-methoxyquinolin-3-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{[4-(dimethylamino)oxan-4-yl]methyl}-1H-pyrazole-4-carboxamide
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(3-chloro-4-fluorophenyl)-4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepane-1-carboxamide