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(5-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}furan-2-yl)methanol
N-cyclopropyl-1-{1-[(2-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
7-(5-chloropyridin-2-yl)-4-(1,4-dioxane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3-{2-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
methyl 4-oxo-4-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butanoate
(3S,4R)-4-(3-methoxyphenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxylic acid
1-(2,3-dihydro-1H-inden-2-yl)-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
1-(3-methylbutyl)-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
13-(6-ethoxy-2,3-dihydro-1H-inden-5-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-methylazepane-2-carboxamide
N'-(adamantan-1-yl)-N-(1H-imidazol-2-ylmethyl)propanediamide
2-(3-fluorophenoxymethyl)-N-methyl-N-(pyrazin-2-ylmethyl)-1,3-oxazole-4-carboxamide
(1R,5R)-3-methanesulfonyl-6-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
1-(2-methylpropyl)-4-oxo-N3-(propan-2-yl)-N5-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-ol
1-[(4-methylphenyl)amino]-N-[(1-methylpiperidin-3-yl)methyl]cyclopentane-1-carboxamide
1-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
3-{[1-ethyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
5-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-3-(2-fluorophenoxy)azetidine
N-[1-(2-phenylethyl)piperidin-3-yl]-3-(1H-1,2,4-triazol-1-yl)propanamide
1-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-N,N-dimethylazepan-4-amine
4-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-fluorophenyl)methyl]piperazin-2-one
6-ethyl-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(morpholin-4-yl)pyrimidin-4-amine
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-methyl-3-(1-methyl-1H-indazol-5-yl)urea
(2S)-4-(methylsulfanyl)-2-{2-[4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}butan-1-ol
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
3-(4-methylphenoxymethyl)-1-(3-phenyl-1,2-oxazole-4-carbonyl)piperidine
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-4,4,4-trifluorobutan-1-one
(2S,4S)-4-amino-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(1,4-dioxan-2-ylmethyl)(methyl){[2-(2-methylphenyl)pyrimidin-5-yl]methyl}amine
N-[1-(3,4,7-trimethyl-1H-indole-2-carbonyl)piperidin-4-yl]pyridin-2-amine
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-cyclooctyl-2-phenylacetamide
N-methyl-2-phenyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
4-({[2-(3,5-dimethoxyphenyl)-2-hydroxyethyl]carbamoyl}amino)-N-ethylbenzamide
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-5-phenylpentan-1-one
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]furan-3-carboxamide
N-{[5-(4-methylphenyl)-1,2-oxazol-3-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
4-{4-[3-(2-chlorophenyl)pyrrolidin-1-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl}pyridine
(3R)-1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidin-3-ol
4-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-6-methyl-1,2-dihydroquinolin-2-one
1-(2-{2-[(3-methoxypyrrolidin-1-yl)methyl]phenoxy}ethyl)-4-methylpiperazine
3-(2-ethylbutyl)-8-(1-methyl-2-oxoimidazolidine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{4-[(2,4-difluorophenyl)methyl]-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(1-ethyl-5-oxopyrrolidin-3-yl)-2-(2-hydroxyphenoxy)acetamide
(4aS,7aR)-1-(2-aminoacetyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[6-(4-fluorophenyl)pyridazin-3-yl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(3S,5R)-1-[(3-ethyl-1H-pyrazol-5-yl)methyl]-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid