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1-methyl-4-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-[1-(benzenesulfonyl)piperidin-4-yl]-2,4-dimethylpyrimidine-5-carboxamide
9-(1,2,4-oxadiazol-3-ylmethyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]propan-1-one
5-{1-[(2,6-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(thiophen-2-ylmethyl)-1-benzofuran-2-carboxamide
N-(2-methyl-1-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}propyl)acetamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}propanamide
2-methyl-7-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decane
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-phenyl-1H-imidazole-5-carboxamide
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]pyridine-2-carbonitrile
N-[3-(dimethylamino)propyl]-N,2,3,5-tetramethylpyrazolo[1,5-a]pyrimidin-7-amine
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
7-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-{[1-(phenoxymethyl)cyclopropyl]methyl}oxolane-2-carboxamide
1-({[1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
N-cyclopentyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2,3-dimethyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}quinoxaline-6-carboxamide
3-hydroxy-3-{1-oxa-7-azaspiro[3.5]nonan-7-ylmethyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-(2-phenylethyl)-5-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,3-benzoxazole
ethyl 4-[5-(morpholin-4-ylmethyl)furan-3-amido]piperidine-1-carboxylate
ethyl 6-methyl-2-({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)pyrimidine-4-carboxylate
5-[4-(morpholine-4-carbonyl)pyridin-2-yl]pyridin-2-amine
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-4-(furan-2-yl)pyrimidine
methyl 2-(3-carbamoylpropyl)-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
3-[4-(3-methylphenyl)piperazin-1-yl]-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}propanamide
(3S,4R)-3-benzyl-1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-methylpiperidin-4-ol
(1-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-yl)methanol
4-chloro-N-(furan-2-ylmethyl)-N-(prop-2-en-1-yl)-2-propanamidobenzamide
N-[(2,5-difluorophenyl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)acetamide
5-[4-(4-fluorophenyl)piperazin-1-yl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
2-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidine-1-carbonyl}-4H-chromen-4-one
8-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({1-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(pyridin-4-yl)ethan-1-one
3-(3-fluorophenyl)-4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1H-pyrazole
8-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N,5-dimethyl-1H-pyrazole-3-carboxamide
N-tert-butyl-5-chloro-2-{[1-(6-methylpyrimidin-4-yl)piperidin-4-yl]oxy}benzamide
3-(5-methyl-1,3,4-thiadiazol-2-yl)-1-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]urea
9-[(4-fluorophenyl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(3-methoxyphenyl)ethyl]methylamine
2-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
N-[(2-ethoxypyridin-3-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-methyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)furan-2-carboxamide
1-(oxan-4-yl)-4-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidine