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{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
(3S,4R)-1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
[(3S,5R)-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-[(5-methylpyrazin-2-yl)methyl]propanamide
N-methyl-2-phenyl-N-[(2E)-3-phenylprop-2-en-1-yl]imidazo[1,2-a]pyridine-6-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(pyridin-4-yl)acetamide
{2-[4-(4-methylphenoxy)piperidin-1-yl]-2-oxoethyl}urea
3-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-2-methyl-4,5,6,7-tetrahydro-2H-indazole
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-methyl-N-[(4-phenoxyphenyl)methyl]acetamide
2-(2,5-dioxoimidazolidin-4-yl)-N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}acetamide
6-fluoro-2-{[4-(2-phenylethyl)piperazin-1-yl]methyl}quinolin-4-ol
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-hydroxy-2-methylbenzamide
2-{2-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}(methyl)amino)methyl]phenoxy}ethan-1-ol
2-amino-N-butyl-4-phenyl-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
3,5-difluoro-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]pyridine-2-carboxamide
N-[1-(2,6-dimethylphenoxy)propan-2-yl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
4-(4-methylphenoxy)-1-(2-phenylethyl)piperidine-4-carboxylic acid
N-[(3-fluorophenyl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
4-methyl-2-oxo-5-{4-[1-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridine-3-carbonitrile
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(5-methyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)propanamide
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propan-1-one
1-[2-(cyclopropylmethyl)-4-{[2-(1H-1,2,3-triazol-1-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
5-(oxolan-2-yl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]thiophene-2-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
2-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2S,4S)-4-amino-N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-1-methylpyrrolidine-2-carboxamide
7-chloro-N,N-dimethyl-2-[2-(pyridin-3-yl)pyrimidin-5-yl]quinoline-4-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
ethyl 4-(cyclopropylmethyl)-1-(quinolin-2-ylmethyl)piperidine-4-carboxylate
N-(2-hydroxyethyl)-N-methyl-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-(3,4-dichlorophenyl)-4-[(2,6-dimethoxyphenyl)methyl]morpholine
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)[2-(methylsulfanyl)ethyl]amine
8-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2-{1H-pyrazolo[3,4-b]pyridin-1-yl}phenyl)methanol
N-methyl-N-(1,2-oxazol-3-ylmethyl)-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(3-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]acetamide
1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-N5-(2-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-butyl-N,1-dimethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
6-amino-2-(2-{[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}ethyl)pyrimidin-4-ol
(4aR,7aS)-1-cyclobutanecarbonyl-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3,4-dimethylphenyl)urea
methyl 3-[2-(2,5-difluorophenyl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2S,4S)-4-amino-1-[4-(azepan-1-ylmethyl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(5-{[ethyl(methyl)amino]methyl}-2-methoxyphenoxy)-3-(piperidin-1-yl)propan-2-ol
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-(furan-2-carbonyl)-4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,4-diazepane
8-(2-amino-6-methoxypyrimidin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
[1-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidin-2-yl]methanol