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2-{4-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-2-oxopiperazin-1-yl}benzonitrile
N-[(5-fluoro-2-methylphenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-(phenylamino)pyrimidine-5-carboxamide
1-(2-methoxyethyl)-3-(2-methylphenyl)-3-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}pyrrolidine-2,5-dione
1-[3-(furan-2-yl)benzoyl]-4-(1H-imidazol-2-yl)piperidine
3-ethyl-8-(4-hydroxy-3-methoxybenzoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(4-{[2-(phenylamino)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-(1,4-dioxan-2-ylmethyl)-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2,3-dimethyl-7-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
6-cyclopentyl-1-methyl-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(2-fluorophenyl)-3-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]propanoic acid
N-ethyl-6-methyl-5-[5-(oxolan-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
2-{1-[2-(1H-imidazol-5-yl)ethyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl}pyrazine
dimethyl({[1-methyl-2-(2-methylpropyl)-7-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl]sulfamoyl})amine
1-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}azetidin-3-ol
1-(3-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}propyl)-1H-imidazole
N-cyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)pent-4-enamide
1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-ol
4-{2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-[3-(2-methoxyethyl)-5-[2-(pyridin-4-yl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
5-methyl-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]pyrimidin-4-amine
3-ethyl-4-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-3-methylpiperazin-2-one
1-ethyl-4-{[5-(3-methoxy-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}pyrrolidin-2-one
2-[(3,4-dimethoxyphenyl)methyl]-N-(1-methoxybutan-2-yl)-1,3-benzoxazole-6-carboxamide
methyl 6-({3-tert-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)pyridine-2-carboxylate
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-4-(3-hydroxy-3-methylbutyl)benzamide
2-amino-6-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[1-(pyridin-2-yl)propyl]amine
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-ethyl-1-(oxan-2-ylmethyl)-3-[2-(prop-2-en-1-yloxy)phenyl]urea
1-(1,4-dioxan-2-ylmethyl)-3-(4-methanesulfonylphenyl)urea
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2,3-dihydro-1-benzofuran-5-carboxamide
1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
4-benzyl-3-ethyl-1-(5-propyl-1,2-oxazole-3-carbonyl)-1,4-diazepan-5-one
N-[1-(2,4-difluorophenyl)ethyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
methyl 2-{4-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
7-(cyclopent-1-ene-1-carbonyl)-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
5-[4-(cyclopentylmethyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
2-(dimethylamino)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(3-methylphenyl)-N-(2-methylpropyl)acetamide
(1R,7S)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-(3-methylbutyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(1-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-yl)(phenyl)methanol
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
3-[2-(2-ethoxyphenoxy)ethyl]-5-methyl-5-(piperidin-4-yl)imidazolidine-2,4-dione
6-methyl-5-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carbonyl}-2-oxo-1,2-dihydropyridine-3-carbonitrile
N-[(4-sulfamoylphenyl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-methyl-9-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[1-(cyclohex-3-en-1-ylmethyl)-4-hydroxypiperidin-4-yl]-N-(thiophen-2-ylmethyl)-1-benzofuran-2-carboxamide