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2-[(4-methoxyphenyl)methyl]-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
5-benzyl-2-methyl-4-{1-[4-(propan-2-yloxy)benzoyl]piperidin-3-yl}pyrimidine
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
N-[(3S)-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
(1R,3S)-3-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)cyclopentane-1-carboxylic acid
8-(1-benzofuran-5-ylmethyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(2-methoxybenzoyl)piperazine
ethyl({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl})(2-methylprop-2-en-1-yl)amine
1-(3,4-dimethoxyphenyl)-2-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethan-1-amine
5-(6-methoxypyridin-3-yl)-4-(4-methylphenyl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
1-[(4-methoxyphenyl)methyl]-4-(oxane-4-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-(3-fluorophenyl)-3-(1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
(2S,4R)-4-(dimethylamino)-1-(2,2-dimethylpropyl)pyrrolidine-2-carboxylic acid
(1R,2R,4R)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-cyclopropyl-1-[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]piperidine-4-carboxamide
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)(methyl)[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amine
1-(2-chloro-6-fluorophenyl)-2-cyclopentanecarbonyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
6-[1-(9H-fluoren-2-ylmethyl)piperidin-4-yl]-2-methyl-3,4-dihydropyrimidin-4-one
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(2-methoxyphenyl)methyl]amine
2-cyclopropyl-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)pyrimidine-5-carboxamide
4-(1-cyclopentyl-5-oxopyrrolidine-3-carbonyl)-1-(4-methylphenyl)piperazin-2-one
1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]urea
5-{4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
2-[4-({ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(5-fluoro-2-methoxybenzoyl)piperidine
2-chloro-N-[(1-ethyl-1H-imidazol-5-yl)methyl]pyridine-4-carboxamide
4-(2-ethylphenyl)-3-[2-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methoxy}acetamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
4-(1H-imidazol-2-yl)-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine
N-[5-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyrimidin-2-yl]benzenesulfonamide
N-cyclopropyl-1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
4-{4-[(2,4-difluorophenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-4-phenylpiperidine-4-carbonitrile
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(2-methylpropyl)piperidin-4-ol
2-[1-(2-methylpropyl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-2-yl]ethan-1-ol
N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carboxamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-4-(piperidin-3-yl)benzamide
2-({2-[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)carbamoyl]phenyl}amino)acetic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
benzyl({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
2-{4-[4-(hydroxymethyl)phenyl]-3,5-dimethyl-1H-pyrazol-1-yl}-N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
2-{1-cyclohexyl-4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-chloro-N-[3-(4-ethoxyphenyl)propyl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
N-methyl-3-(2-methylphenyl)-N-(1-methylpiperidin-4-yl)-3-phenylpropanamide
7-methyl-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide