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(3aS,6aS)-2-(cyclopent-3-ene-1-carbonyl)-5-(pyridin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
1-[(4-chlorophenyl)methyl]-N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
3-{[1-(azepane-1-sulfonyl)pyrrolidin-3-yl]methyl}benzamide
3-{[(2H-1,3-benzodioxol-5-ylmethyl)amino]methyl}-1-(2-methoxyethyl)-6-methyl-1,2-dihydroquinolin-2-one
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-methoxybenzamide
ethyl 1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-3-(2-phenylethyl)piperidine-3-carboxylate
4-[(4-fluorophenyl)methyl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
2-methyl-4-{1-[(3-phenyloxolan-3-yl)methyl]piperidin-4-yl}pyrimidine
4-[2-(methoxymethyl)pyrimidin-5-yl]-3-methyl-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
4-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-phenyl-1H-pyrazole
N-methyl-N-(1,3-thiazol-2-ylmethyl)-4-(1H-1,2,4-triazol-1-yl)butanamide
1-(oxan-4-yl)-4-[2-(2-phenylethynyl)phenyl]-1H-1,2,3-triazole
2-amino-4-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-methyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)pyrrolidin-2-yl]-1-methyl-1H-1,3-benzodiazole
1-(dimethylsulfamoyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
(4aR,8aS)-1-butyl-6-[(5-methylfuran-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
4-fluoro-3-(4-fluoropiperidine-1-carbonyl)benzene-1-sulfonamide
(1S,5R)-6-benzyl-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(oxan-2-ylmethyl)-1,2,3,4-tetrahydroquinolin-2-one
4-[5-(4-acetylphenoxymethyl)-1,2-oxazole-3-carbonyl]-1-cyclopentylpiperazin-2-one
N-benzyl{[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]amino}sulfonamide
2-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]-6-phenyl-3,4-dihydropyrimidin-4-one
2-benzyl-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1,3-thiazole-4-carboxamide
2-ethyl-9-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(2-ethoxyphenyl)methyl]-N,2-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[3-(4,4-diphenylpiperidin-1-yl)-3-oxopropyl]pyrrolidin-2-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-4-methyl-1H-imidazole-5-carboxamide
(3S,5R)-N3-cyclopropyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,1,3,7-tetramethyl-1H-indole-2-carboxamide
(3aR,7aS)-N-[3-(1H-pyrazol-1-yl)phenyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
1-phenyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-chloro-N-{[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-3-yl]methyl}benzamide
8-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-3-ol
2-(2-aminoethyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}quinazolin-4-amine
2-(3-{[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl}phenoxy)acetic acid
5-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}-2-(furan-2-yl)pyrimidine
N-{1-[4-(4-methoxybenzoyl)piperazin-1-yl]-1-oxopropan-2-yl}methanesulfonamide
(4aS,8aR)-1-(3-aminopropyl)-6-(1-benzofuran-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(4,4,4-trifluorobutyl)-2,7-diazaspiro[4.5]decane
2-methoxy-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-N-ethylpiperidine-1-carboxamide
(2S,4S)-4-(benzylamino)-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
4-(4-chlorophenoxy)-N-[3-(pyridin-4-yl)propyl]piperidine-4-carboxamide
1-(5-chloro-2-methylphenyl)-3-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)propan-1-one
2-[2-(2-methyl-1,4-oxazepan-4-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
2-[2-benzyl-5-oxo-4-(3-phenylphenyl)piperazin-1-yl]acetamide