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4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[3-(methylsulfanyl)propyl]piperidine
2-ethyl-8-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-N,N-diethyl-1-(3-oxo-3,4-dihydroquinoxaline-2-carbonyl)pyrrolidine-2-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(oxolane-2-carbonyl)-1,4-diazepane
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-fluoro-6-methoxy-N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)benzamide
4-{1-[4-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazol-2-yl}benzene-1,2-diol
ethyl 4-[(3-fluorophenyl)methyl]-1-(oxane-4-carbonyl)piperidine-4-carboxylate
(1S,5R)-6-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-phenyl-1-(pyridin-3-ylmethyl)piperidin-4-yl]ethan-1-one
N-[(4-ethylphenyl)methyl]-N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N2-[cyclopropyl(6-methylpyridin-2-yl)methyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-cycloheptylpiperidin-3-yl)-3-(2-oxoimidazolidin-1-yl)benzamide
5-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-tert-butyl-4-hydroxy-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}pyrimidine-5-carboxamide
1-(4-methoxyphenyl)-3-(2-methylpropyl)-5-(1H-pyrazol-1-ylmethyl)-1H-1,2,4-triazole
1-(4-chlorophenyl)-2-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethan-1-ol
methyl 1-methyl-3-(3-phenylpropanamido)-5-[(thiolan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-(butan-2-yl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
5-[(1-benzothiophen-2-ylmethyl)amino]-1-methyl-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2E)-1-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]-3-(pyridin-3-yl)prop-2-en-1-one
5-methoxy-2-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}-3-methyl-1H-indole
2-{2-[(1S,5S)-3-azabicyclo[3.3.1]nonan-3-yl]-2-oxoethyl}-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
N-ethyl-6-methoxy-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(3-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
4-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]pyridine
[(1r,4r)-4-{[(6-ethylpyrimidin-4-yl)amino]methyl}cyclohexyl]methanol
1-[(4aR,8aR)-4a-hydroxy-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-2-yl]-3-(1H-pyrazol-1-yl)propan-1-one
1-[(4-cyanophenyl)methyl]-4-(4-methylphenoxy)piperidine-4-carboxylic acid
methyl 6-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)pyridine-2-carboxylate
2-(dimethylamino)-2-(4-fluorophenyl)-N-[1-(oxan-4-yl)piperidin-4-yl]acetamide
7-fluoro-N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-3-methyl-1H-indole-2-carboxamide
2-{pyrazolo[1,5-a]pyridin-7-yl}-1,3-thiazole
N-methyl-2-[methyl(2-phenylethyl)amino]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
methyl 2-(4-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-oxopiperazin-1-yl)acetate
6-[({1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}amino)methyl]-1,4-oxazepan-6-ol
5-(2,4-difluorophenoxymethyl)-N-(1H-indol-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-{1-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]piperidin-3-yl}benzoic acid
1-methyl-1'-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-[1-(4-fluorophenyl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[2-(ethanesulfonyl)ethyl]-1,3-benzothiazole-6-carboxamide
2-methyl-6-(propan-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrimidin-4-amine
N-[3-(azepan-1-yl)-2-hydroxypropyl]-2-fluoro-5-sulfamoylbenzamide
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3,5-dimethyl-2-{[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}-1,4-dihydropyridin-4-one
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanamide
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-propoxypropan-1-one