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3-(2-chlorophenyl)-1-cyclopentyl-3-{2-[4-(1-hydroxypropyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
1-(3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-oxopropyl)azepan-2-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[5-(propan-2-yl)thiophene-3-carbonyl]pyrrolidin-3-yl]methanol
N,1,3-trimethyl-N-(1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-2-phenylethyl)-1H-pyrazole-5-carboxamide
2-ethoxy-1-[1-(hydroxymethyl)-9-(pyridin-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
1-{4-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-2-(1H-imidazol-4-yl)ethan-1-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
N-[4-(2,2-dimethylpropanamido)-3-methylphenyl]-2,4-dimethoxybenzamide
(1R,7S)-3-[4-(2-hydroxyethyl)phenyl]-N-methyl-4-oxo-N-(pyrazin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-methyl-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
5-fluoro-2-(2-fluoro-3-methoxyphenyl)pyridine
4-(5-ethylpyrimidin-2-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-(2-methoxyethyl)-1-methyl-6-oxo-N-(thiophen-2-ylmethyl)-1,6-dihydropyridine-3-carboxamide
(2S,4R)-1-methyl-4-[2-(4-phenylphenyl)acetamido]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(4-fluorophenyl)ethyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-[(3-methylpyridin-2-yl)methyl]propanamide
1-(5-methyl-1,2-oxazole-3-carbonyl)-3-(4-phenylbenzoyl)piperidine
6-(azepan-1-yl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-[3-(1,2-oxazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
methyl({[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})[1-(pyrimidin-4-yl)ethyl]amine
2-(furan-2-yl)-N-methyl-2-oxo-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]acetamide
5-({4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)pentan-1-ol
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-3-(pyrazin-2-yl)propanamide
1-[3-(4,5-dihydro-1H-imidazol-2-yl)phenyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-{2-[methyl(phenyl)amino]propyl}-3-[1-(2-methylpropyl)-1H-pyrazol-5-yl]urea
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-[(3-methoxyphenyl)methyl]-4-(1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
3-{[(2-hydroxyethyl)(propyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-(1-ethoxy-2-methylpropan-2-yl)-3-[(2-fluorophenyl)formamido]propanamide
8-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(5-aminopyridin-3-yl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
1-[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]-2-(3-hydroxyadamantan-1-yl)ethan-1-one
methyl 5-{4-[5-(2-methoxy-2-phenylacetamido)-1H-pyrazol-1-yl]piperidin-1-yl}-5-oxopentanoate
1-(4-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
3-(cyclopropylmethyl)-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-3-carboxylic acid
4-(4-chlorophenyl)-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]butanamide
N-(1-{1-[(dimethylcarbamoyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
7,7-dimethyl-2-(2-methyloxolan-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(3S,4R)-1-(5-hydroxypyrazine-2-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
1-(cyclobutylmethyl)-3-hydroxy-3-({[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]amino}methyl)piperidin-2-one
1-(2-{[(3-methylphenyl)methyl]amino}ethyl)-N-phenyl-1H-1,2,3-triazole-4-carboxamide
2-cyclopropyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1,3-benzoxazole-6-carboxamide
3-[1-(3-propyl-1,2,4-oxadiazol-5-yl)ethyl]-3,4-dihydroquinazolin-4-one
(1S,5R)-6-(pyridin-2-ylmethyl)-3-(1,3-thiazol-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one