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4-[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(2,4-difluorophenyl)-3-{1-oxaspiro[4.4]nonan-3-yl}urea
2-(methylamino)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1,3-thiazole-4-carboxamide
2-chloro-5-{[4-(4-fluoro-3-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
ethyl 5-(1H-indol-3-ylmethyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[2-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-6-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
5-{2-[1-(propan-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}-1H-1,2,3-benzotriazole
ethyl 1-[(5-chloro-2-methoxyphenyl)carbamoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N-[1-(2-fluorophenyl)piperidin-4-yl]-5,6-dimethylpyrimidin-4-amine
1-benzyl-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-chloro-4-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]benzamide
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
3-chloro-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-ethyl-N-methylpyrimidine-5-carboxamide
4-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidine-1-carbonyl]-1λ6-thiane-1,1-dione
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-[1-(5-phenyl-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
(3S,5R)-1-ethyl-5-[(4-fluorophenyl)carbamoyl]piperidine-3-carboxylic acid
N-[2-(4-fluorophenoxy)ethyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)(4,4,4-trifluorobutyl)amine
1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-N-methylpyrrolidine-3-carboxamide
N-[1-(oxan-4-yl)piperidin-4-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
N-[4-(4-{[(2-methylphenyl)(pyridin-4-yl)methyl]amino}piperidin-1-yl)phenyl]pyrazine-2-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
3-{[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-4-(2-phenylethyl)-4H-1,2,4-triazole
2-(3-methylbut-2-en-1-yl)-8-[2-(phenylsulfanyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-[1-cyclopentyl-4-(2,3-dihydro-1H-inden-2-yl)piperazin-2-yl]ethan-1-ol
9-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1S,2R)-2-aminocyclobutyl]-2-methyl-5-[5-(trifluoromethyl)-1H-pyrazol-3-yl]furan-3-sulfonamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(oxan-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[(1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)methyl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2-(2-phenylethyl)morpholine
2-phenyl-5-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-2,3-dihydro-1H-pyrazol-3-one
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
(4aR,7aS)-1-(3-methylbutanoyl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-3-(2-oxopyrrolidin-1-yl)propanamide
2-ethyl-1-({4-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}methyl)-1H-imidazole
N-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-3-(1H-pyrazol-4-yl)benzamide
ethyl 4-{1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}piperazine-1-carboxylate
(1S,6R)-3-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-3,9-diazabicyclo[4.2.1]nonane
N-[(1S,2R)-2-aminocyclobutyl]-1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carboxamide
(3S,4S)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methylacetamide
5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-1-(2-methoxyphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
5-(2,6-difluorophenoxymethyl)-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-1,2-oxazole-3-carboxamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(4aR,8aR)-4-[(2-fluoro-4-methoxyphenyl)methyl]-octahydro-2H-1,4-benzoxazine
4-[(2R,3S,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butanoic acid
3-[2-(4-methyl-3-oxopiperazin-1-yl)-2-oxoethyl]-3,4-dihydroquinazolin-4-one
4-{1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}thiomorpholine