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(3S,4R)-3-methoxy-1-(5-phenyl-1H-pyrrole-2-carbonyl)piperidin-4-amine
3-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
4-({4-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]furan-2-yl}methyl)morpholine
1-(2,3-dihydro-1H-inden-2-yl)-5-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazol-5-yl]-1H-1,2,4-triazole
N-(1-benzyl-1H-pyrazol-5-yl)-2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
3-({3-[cyclopentyl(methyl)amino]propyl}carbamoyl)benzoic acid
3-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-3H,4H-pyrido[2,3-d]pyrimidin-4-one
4-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-N-methylpyridin-2-amine
N-[(2R,4R,6S)-2-(propan-2-yl)-6-[3-(pyridin-2-ylmethoxy)phenyl]oxan-4-yl]acetamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]acetamide
2-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(4-chloro-2-methoxy-5-methylphenyl)-3-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-3-methylurea
2-{4-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-ylmethyl]-2-chlorophenoxy}acetamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(4-cyano-5-methyl-1H-pyrrol-2-yl)methyl]piperidine-4-carboxylic acid
6-(8-methoxy-2-methylquinolin-5-yl)-9H-purin-2-amine
4,6-dimethyl-2-{[2-(3-methyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]methyl}pyrimidine
methyl (1R,3S,3aR,6aS)-5-benzyl-3-(4-fluoro-2-hydroxyphenyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-(2-methyl-1,3-thiazol-4-yl)-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
6-methoxy-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[4-(3-chlorophenyl)piperazin-1-yl]-6-ethyl-5-methylpyrimidin-2-amine
3-benzyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
[1-({[2-(dimethylamino)-6-methylpyrimidin-4-yl](methyl)amino}methyl)cyclobutyl]methanol
3-[benzyl({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amino]-2-methylpropan-1-ol
4-{1-[4-(furan-2-yl)benzoyl]piperidin-3-yl}-5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidine
6-(3-benzyl-1H-1,2,4-triazol-5-yl)-1,3-benzothiazole
8-[(4-hydroxyphenyl)methyl]-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1,3-dimethyl-8-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,3R,6R)-5-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-chloro-4,6-dimethyl-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-[3-(methylsulfanyl)phenyl]ethan-1-one
2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]acetic acid
5-(azepane-1-carbonyl)-N-[(2,4-difluorophenyl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(2-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}phenoxy)acetic acid
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-{3-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-3-oxopropyl}-N-methylmethanesulfonamide
2-[(3,5-difluorophenyl)methyl]-8-[3-(methylsulfanyl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
1-({3-[3-(diethylamino)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)-1,4-diazepan-5-one
N-(2,4-dimethylpentan-3-yl)-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-7-fluoro-N,3-dimethyl-1H-indole-2-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(1-propylpiperidin-4-yl)acetamide
ethyl 1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-pyrazole-4-carboxylate
6-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}-2-oxo-N-[1-(thiophen-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
5-(4-methoxyphenyl)-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}furan-2-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}acetamide
5-{[4-(4-methoxyphenoxy)piperidin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
3-(2-methylphenyl)-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
N-methyl-2-{4-oxo-6-phenyl-3H,4H-thieno[2,3-d]pyrimidin-3-yl}acetamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
methyl 3-cyclohexaneamido-6-(piperidin-1-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
2-ethyl-9-[4-(1,3-oxazol-5-yl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one