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methyl 2-[(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)methyl]-1,3-oxazole-4-carboxylate
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-3-(piperidin-4-ylmethyl)benzamide
3-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]benzoic acid
3-hydroxy-1-(2-methoxyethyl)-3-[(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)methyl]piperidin-2-one
2-(dimethyl-1,2-oxazol-4-yl)-N-[(dimethyl-1,3-thiazol-2-yl)methyl]acetamide
(3aR,6aR)-2-acetyl-5-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-1-propyl-N-[2-(pyridin-2-yl)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
9-[(2S)-2-hydroxy-2-phenylacetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-4-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-(pyridin-4-yl)quinoline
(1R,3S,5S)-8-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-8-azabicyclo[3.2.1]octan-3-ol
4-methyl-5-[2-(2-phenylethyl)piperidine-1-carbonyl]pyrimidine
3-[2-(1-ethylpiperidin-4-yl)acetamido]-3-(naphthalen-1-yl)propanoic acid
(3S,7S)-5-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-(dimethylamino)-8-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
ethyl 2-[methyl({5-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]pyrimidin-2-yl})amino]acetate
(1R,7S)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-3-(2-phenoxyethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-(furan-2-ylmethyl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
N-{[1-(2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}acetyl)piperidin-3-yl]methyl}acetamide
2-{4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carboxamide
N,8-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
5-chloro-3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
2-[(5-methylpyrazin-2-yl)methyl]-9-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
4-cyclobutaneamido-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
1-cyclopentyl-N-[2-(methylsulfanyl)ethyl]-6-oxopiperidine-3-carboxamide
methyl (2S,3S)-2-[(2-benzyl-1-methyl-5-propanamido-1H-1,3-benzodiazol-7-yl)formamido]-3-methylpentanoate
(2S,4S)-4-{[(2,6-difluorophenyl)methyl]amino}-1-(naphthalen-1-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(1R,2R)-N-(2-methoxyethyl)-2-phenyl-N-(thiophen-2-ylmethyl)cyclopropane-1-carboxamide
2-fluoro-6-hydroxy-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)benzamide
4-({[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]amino}methyl)-2,6-dimethylphenyl acetate
5-fluoro-N4,N4-dimethyl-N2-[(3-phenyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4-diamine
(3S,4R)-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-4-(3-methylthiophen-2-yl)piperidin-3-ol
3-[(3R,4S)-4-(dimethylamino)-1-[2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetyl]piperidin-3-yl]propanoic acid
1-(1-benzylpiperidine-2-carbonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
(2S,4S)-4-amino-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-N-methylpyrrolidine-2-carboxamide
1-cyclohexyl-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1-propyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-(2-hydroxyethyl)-N-methyl-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carboxamide
3-(2-hydroxyphenyl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
9-hydroxy-2-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
(3R,4R)-1-[(2,3-dichloro-6-fluorophenyl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
6-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purin-2-amine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3-chlorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(piperidin-1-yl)ethyl]amino}methyl)piperidin-2-one
[5-(1-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-imidazol-2-yl)furan-2-yl]methanol
1-(5-propyl-1,2-oxazole-3-carbonyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine