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1'-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-[1-(1-methylpiperidine-4-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-cyclohexyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-4-carboxamide
N-benzyl-3-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]benzamide
3-[(3-chlorophenyl)methyl]-1-(pyrazin-2-yl)piperidine-3-carboxylic acid
(5S,9aS,9bS)-5-(8-methoxy-2H-chromen-3-yl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1,5-dimethyl-4-{[3-(2-methylphenyl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazine
N-[2-(azepan-1-yl)-2-phenylethyl]-1-methanesulfonylpiperidin-4-amine
N-[(3,4-difluorophenyl)methyl]-3-{1-[2-(pyridin-3-yl)acetyl]piperidin-3-yl}propanamide
2-[2-(3,4-dichlorophenyl)morpholin-4-yl]quinoxaline
2-{3-cyclopropyl-5-[2-(4-phenylphenyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-(2-methoxy-4-methylphenoxymethyl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
3-cyclopropyl-5-(2,2,2-trifluoro-1-methoxy-1-phenylethyl)-1H-1,2,4-triazole
4-{2-[(dimethylamino)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-1,3-dimethyl-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid
benzyl({[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl})methylamine
(2R,3R,6R)-5-(1H-1,3-benzodiazol-2-ylmethyl)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(4-chlorophenyl)-1-[3-(morpholin-4-yl)azetidin-1-yl]-3-phenylpropan-1-one
2-({4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
2-{3-[hydroxy(phenyl)methyl]-1-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethan-1-ol
[3-(2-chloro-6-methoxyphenyl)-4-fluorophenyl]methanamine
3-cyclopropyl-6-[(3,5-dimethoxyphenyl)methyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-[2-({methyl[(1-methylpyrrolidin-2-yl)methyl]amino}methyl)-4-(pyrazin-2-yl)phenoxy]acetic acid
2-chloro-5-{1-[2-(4-methyl-1H-pyrazol-1-yl)propyl]-4-phenyl-1H-imidazol-5-yl}pyridine
(3S,4S)-1-[benzyl(methyl)sulfamoyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-(thiophen-3-ylmethyl)piperidine
1-(diphenylmethyl)-4-(piperidin-3-ylmethyl)piperazine
5,5-dimethyl-3-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-1,3-oxazolidine-2,4-dione
4-phenoxy-1-(thiophene-2-carbonyl)piperidine-4-carboxylic acid
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carboxamide
1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-1,4-diazepane
2-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
(4aS,7aR)-1-butanoyl-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-chlorophenoxy)-1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(methylsulfanyl)acetamide
2-{1-cyclopentyl-4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
3-methyl-1-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}urea
6-(4-tert-butylbenzoyl)-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-3-phenylpyrrolidin-3-ol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-methyl-1H-1,3-benzodiazole-2-carboxamide
N-{[2-(4-chlorophenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-3-carboxamide
N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
(4aS,8aR)-6-(2,1-benzoxazole-3-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
(1R,5R)-6-[(1-methyl-1H-indol-2-yl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-(furan-2-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(3-methyl-1H-pyrazol-5-yl)methyl]amine
1-methyl-3-propyl-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-pyrazole
7-(2-cyclohexylethyl)-2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2,7-diazaspiro[4.5]decane
2-(2-aminoethyl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)quinazolin-4-amine
3-({2-[(4-fluorophenyl)methyl]morpholin-4-yl}methyl)-1H-indole