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2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}ethan-1-one
N-[(3R,4S)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
5-methyl-6-(2-methylpiperidine-1-carbonyl)-N-[(4-phenyloxan-4-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
2-hydroxy-2-(4-methoxyphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]amino}methyl)piperidin-2-one
3-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylpropanamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-5-methyl-1H-indazole-3-carboxamide
6-[3-(3-methylphenyl)benzoyl]-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(pyridin-4-yl)propan-1-one
2-(1-methylpiperidin-2-yl)-1-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethan-1-one
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(oxan-4-yl)acetamide
2-(4-{[(3S)-3-(dimethylamino)azepan-1-yl]methyl}phenoxy)ethan-1-ol
1-(4-benzylpiperazin-1-yl)-3-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]propan-1-one
1-[2-(3-chlorophenyl)ethyl]-4-[(1H-imidazol-4-ylmethyl)amino]pyrrolidin-2-one
7-fluoro-N-methyl-N-(oxan-2-ylmethyl)quinazolin-4-amine
5-(3,4-difluorophenoxymethyl)-3-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1,2-oxazole
2-(morpholin-3-yl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)acetamide
[(2-butyl-1H-imidazol-4-yl)methyl](methyl){[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[(2-chlorophenyl)methyl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-(4-fluorophenyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]cyclopropane-1-carboxamide
[2-(3-methoxyphenyl)-1-[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]ethyl](methyl)(pyridin-4-ylmethyl)amine
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-[4-(furan-2-ylmethoxy)phenyl]urea
N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(1-benzofuran-2-ylmethyl)-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-methyl-7-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(3,4,5-trimethoxyphenyl)acetamide
methyl 2-oxo-8-(3-phenylbutyl)-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
4-(4-{[3-(furan-2-yl)-3-phenylpropyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
5-(2-chloro-4-fluorobenzoyl)-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]-2-phenylethan-1-ol
3-(3-methoxyphenyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-pyrazole-4-carboxamide
(1R,5R)-3-(4-cyclopentylpyrimidin-2-yl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
6-methyl-5-{2-oxo-2-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3R,4R)-1-(1-benzoxepine-4-carbonyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-ethyl-N-[(2-methoxyphenyl)methyl]-6-methylpyrimidin-4-amine
8-[6-(dimethylcarbamoyl)pyrazin-2-yl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(propan-2-yl)-2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylformamido)acetamide
N-[3-(2,6-dimethylphenoxy)propyl]-N,2,4-trimethyl-1,3-thiazole-5-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(1H-imidazol-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-({[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]carbamoyl}amino)-4-methoxy-N-methylbenzamide
2-(cyclopropylmethyl)-8-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-ethyl-2-{1-[2-(pyridin-3-yl)ethyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
4-(2-methoxyquinolin-3-yl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
(2-{8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)urea
8-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,N-diethyl-1-[(1s,4s)-4-(2,5-dimethoxybenzenesulfonamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-(1-benzothiophene-5-carbonyl)-3-(3-fluorophenyl)piperazin-2-one
6-[3-(4-methoxyphenoxymethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[(1r,4r)-4-hydroxycyclohexyl]amino}methyl)piperidin-2-one