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2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-[3-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
1-cyclopropanecarbonyl-4-({4-[3-(furan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-3-yl]methanol
methyl[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl][(5-methyl-1H-pyrazol-3-yl)methyl]amine
2-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-N-methylacetamide
2-{4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
2-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
5-[4-(1,2-benzothiazol-3-yl)piperazine-1-carbonyl]pyrazin-2-ol
1-[1'-(2,3-dihydro-1-benzofuran-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-methyl-3-(2-methylpropyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
2-{2-[(3-methoxyphenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetamide
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-cyclohexyl-N-methylacetamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
(2S,4R)-N-methyl-1-(1-propylpiperidin-4-yl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-{2-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]ethyl}pyridine-3-carboxamide
3-(4-hydroxyphenyl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-5-carboxamide
5,5-diphenyl-1-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}piperidin-2-one
N-cyclopentyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-[4-(3-fluorophenyl)phenyl]-1-(pyridine-3-carbonyl)pyrrolidine-2-carboxamide
5-cyclobutanecarbonyl-1'-(5-methylpyrazine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(3,3,3-trifluoropropyl)pyrimidine
8-(2-amino-6-methylpyrimidine-4-carbonyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-benzyl-N-(3-hydroxy-2-methylpropyl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
6-{[1-(morpholin-4-yl)hex-5-en-2-yl]oxy}pyridine-2-carbonitrile
2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carboxamide
N-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
(7R,9aR)-N-(3-fluorophenyl)-6,9-dioxo-7-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(3-methoxypropyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{4-[(3-ethoxy-4-methoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
4-(3,4-difluorobenzenesulfonyl)-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-5-methyl-1,2-oxazole-4-carboxamide
N-methyl-N-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-2,3-dihydro-1H-inden-2-amine
2-ethyl-8-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
methyl (1R,5S,6R)-6-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)-3-azabicyclo[3.1.0]hexane-3-carboxylate
N-[2-(quinolin-3-yl)pyridin-3-yl]cyclopropanecarboxamide
1-(1-methylpiperidine-2-carbonyl)-4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
[(4-{2-[4-(benzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
methyl 2-{[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]methyl}-1,3-oxazole-4-carboxylate
N-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-propyl-1H-pyrazole-4-carboxamide
1,1-dioxo-N-[2-(propylsulfanyl)phenyl]-1λ6-thiomorpholine-4-carboxamide
dimethyl[2-(2-{1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
2-[1-(5-chloro-2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyrazine
3-(4-phenyl-1H-pyrazol-5-yl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
4-[(4-chlorophenyl)methyl]-3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(pyridin-3-yl)ethan-1-one
2-(1-tert-butyl-1H-pyrazol-4-yl)-6-ethyl-N,N-dimethylquinoline-4-carboxamide