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7-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
3-(3-fluorophenyl)-6-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
ethyl 1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazole-2-carboxylate
1-[(3,4-dimethoxyphenyl)methyl]-4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]piperidine
2-[4-(4-fluorophenyl)butanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[1'-(trimethyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
5-[2-(3,4-dimethoxyphenyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-(isoquinolin-5-yl)-N,N,1-trimethyl-1H-1,2,4-triazol-5-amine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-phenoxypropanamide
2-methyl-6-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
2-(3,4-dimethoxyphenyl)-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-3-(dimethylsulfamoyl)-5-[(thiophen-3-ylmethyl)amino]benzamide
1'-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
1-{[1-(2H-1,3-benzodioxol-5-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-2-one
11-{methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
4-[(3-methyl-1,2-oxazol-5-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}-N-propylaniline
1-{4-[(5-fluoro-2-methylphenyl)methyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
2-[(3R,4S)-3-[2-(3-fluorophenoxy)acetamido]-4-(propan-2-yl)pyrrolidin-1-yl]acetic acid
5-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidine-1-carbonyl)pyrazin-2-ol
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N1,N1-dimethyl-N3-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)piperidine-1,3-dicarboxamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
2-butyl-N-(1-propyl-1H-1,2,3-triazol-4-yl)-2,5-dihydro-1H-pyrrole-1-carboxamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-{[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}-N-(4-methylphenyl)propanamide
1-(3-methoxyphenyl)-4-[2-(methylamino)pyridine-4-carbonyl]piperazin-2-one
2-(2-chloro-4-{[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]methyl}phenoxy)acetamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(4-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-(3-methyl-1H-pyrazole-5-amido)-N-phenylpiperidine-1-carboxamide
1-[4-methyl-2-({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)pyrimidin-5-yl]ethan-1-one
3-(5-{1-[(1S)-2,3-dihydro-1H-inden-1-yl]-1H-imidazol-2-yl}thiophen-3-yl)prop-2-yn-1-ol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
3-{5-[2-(4-methylbenzoyl)phenyl]-1,2,4-oxadiazol-3-yl}pyridazine
2-[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indole
N-cyclohexyl-2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]acetamide
1-benzyl-8-(1H-indol-3-ylmethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N5-benzyl-N6-[1-(1,3-thiazol-2-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-1-(4-methylphenyl)piperazin-2-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-(pyrrolidin-3-yl)benzamide
1'-(1-ethyl-1H-pyrazole-5-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
9-methoxy-7-[4-(methylsulfanyl)phenyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(1H-pyrazol-1-ylmethyl)piperidine
2-(2-{[4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
N-{[7-(2,2-dimethyloxane-4-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
1-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-pyrazole-5-carboxamide
3-fluoro-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-{3-[3-(3-ethylphenoxy)azetidine-1-carbonyl]piperidin-1-yl}acetamide