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1-(2-methoxyphenyl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
1-methyl-5-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-(1-methoxybutan-2-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
4-(2-{[1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}ethyl)benzene-1-sulfonamide
1-(3,5-dimethylphenyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazin-2-one
methyl (2S,4R)-4-(dimethylamino)-1-(3-methylfuran-2-carbonyl)pyrrolidine-2-carboxylate
N-[(3-hydroxypyrrolidin-3-yl)methyl]-4-methoxy-3-(morpholin-4-yl)benzamide
4-{5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl}pyridine
3-methyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
2-[4-(4-hydroxy-4-phenylpiperidine-1-carbonyl)phenoxy]acetamide
2-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-azaspiro[4.4]nonan-3-one
(1S,5R)-6-benzyl-3-{[3-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-butyl-3-({[(4-methoxyphenyl)methyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[(4,6-dimethylpyridin-3-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-acetyl-N-[2-(cyclohex-1-en-1-yl)ethyl]-N-[(4-methoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(1-phenyl-1H-pyrazol-4-yl)methyl]amine
4,4,4-trifluoro-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}butanamide
1-(azocan-1-yl)-3-[(3S,4R)-1-(2-methylpropyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-one
4-[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
(3aS,6aS)-2-[(4-chlorophenyl)methyl]-5-cyclobutanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2,4-dichlorophenoxy)-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]acetamide
2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide
N-[3-(4-ethylpiperazin-1-yl)propyl]-6-(methoxymethyl)pyridine-2-carboxamide
1-(cyclohexylmethyl)-3-({[2-(morpholin-4-yl)ethyl]amino}methyl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)[(2,3,6-trifluorophenyl)methyl]amine
3-methyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-(propan-2-yl)piperazine-1-carboxamide
1-ethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(pyrrolidin-1-yl)piperidine
(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}-1,2,3,6-tetrahydropyridine
N-benzyl-1-{2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
1-(difluoromethyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
(1S,5R)-6-(1-benzofuran-2-ylmethyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{2-[(4-chlorophenyl)methoxy]ethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
4-[3-(3-methoxypropyl)piperidin-1-yl]-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
1-(2-{[2-(cyclohex-1-en-1-yl)ethyl]amino}pyrimidin-4-yl)piperidin-4-ol
N-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-3-(1-methyl-1H-pyrazol-4-yl)propanamide
N,N-diethyl-2-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
2-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
5-(methoxymethyl)-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylfuran-2-carboxamide
1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3-(1H-imidazol-2-yl)piperidine
4-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
6-(dimethylamino)-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)pyridine-3-carboxamide
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-(thiophen-3-ylmethyl)piperidin-3-ol
6-[(3-methoxyphenyl)methoxy]-4-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
ethyl 4-{[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]amino}piperidine-1-carboxylate
N,N-dimethyl-2-{methyl[2-(quinolin-4-yloxy)hex-5-en-1-yl]amino}acetamide
4-[2-(pyrazin-2-yloxy)hex-5-en-1-yl]thiomorpholine
2-[(1S,5R)-3-(5-chloro-2-hydroxybenzoyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-[2-chloro-5-(diethylcarbamoyl)phenyl]pyridine-2-carboxamide