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3-(dimethyl-1,2-oxazol-4-yl)-N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}propanamide
3-[({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1λ6-thiolane-1,1-dione
3-{1-[(4-chlorophenyl)methyl]-1H-pyrazol-5-yl}-1-{1-oxaspiro[4.4]nonan-3-yl}urea
N-{1-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]-1H-pyrazol-4-yl}pyridine-2-carboxamide
N-ethyl-5-({3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyrimidin-2-amine
5-chloro-4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}-2-methoxyphenol
N-[(4-cyanophenyl)methyl]-3-methoxy-2,2-dimethylpropanamide
2-(5-acetylthiophen-3-yl)-N,N-bis(1,3-oxazol-4-ylmethyl)acetamide
(1S,5R)-3-cyclobutanecarbonyl-6-[5-(methoxymethyl)thiophene-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
(5-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazine-1-carbonyl}furan-2-yl)methanol
4-[(2,4-difluorophenyl)methyl]-7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-3-phenylpiperazine
1-(1-{imidazo[1,2-a]pyridine-6-carbonyl}piperidin-4-yl)-3-phenylpropan-1-ol
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl 4-{[(1,1-dioxo-1λ6-thiolan-3-yl)(ethyl)amino]methyl}benzoate
1-[(4,5-dimethylfuran-2-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-2-phenoxy-N-(pyridin-3-ylmethyl)acetamide
N-(3-phenylphenyl)-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
1-{2-[5-(2-hydroxy-6-methylpyridin-4-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrrolidin-2-one
N-[(2-fluorophenyl)methyl]-3-{1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}propanamide
1-[2-(dimethylamino)-4-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl){[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}amine
4-methyl-1-[2-(4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazol-1-yl)ethyl]-1H-1,2,3-triazole
2-{2-[1-(cyclopent-3-en-1-yl)-4-phenyl-1H-imidazol-5-yl]phenoxy}ethan-1-ol
N-methyl-2-(4-{[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyrimidin-4-amine
N-{[1-(1H-indol-2-ylmethyl)pyrrolidin-3-yl]methyl}-2-(1H-pyrazol-1-yl)acetamide
ethyl 1-(2,3-dihydroxypropyl)-4-[(3-fluorophenyl)methyl]piperidine-4-carboxylate
1-{3-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}azepane
N-(4-hydroxybutyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-[2-(benzyloxy)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
2-hydroxy-2-(4-methoxyphenyl)-1-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
N-({7-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)methanesulfonamide
methyl (2S,4R)-4-[(phenylcarbamoyl)amino]-1-(3-phenylpropyl)pyrrolidine-2-carboxylate
(4S,6R)-N-[3-(2-ethylphenoxy)propyl]-N,6-dimethyl-2-sulfanylidene-1,3-diazinane-4-carboxamide
1-(4-{[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
2-[1-(1-methylpiperidin-4-yl)-4-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
1-[(2-fluorophenyl)methyl]-6-oxo-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
(2R,6R)-4-(2,5-difluorobenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
6-(4-fluorophenyl)-N-methyl-N-(oxan-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
8-[(2-aminopyridin-3-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 5-cyano-2-methyl-6-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyridine-3-carboxylate
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(3S,4R)-4-ethoxyoxolan-3-yl]-1H-1,2,3-triazole
(4aR,7aS)-1-(2-methoxyethyl)-4-(quinolin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(pyridin-2-yl)acetamide
N-cyclopentyl-6-{7-methyl-2,7-diazaspiro[4.4]nonan-2-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine