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2-{[(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
4-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-3-methyl-4H,5H,6H,7H-[1,2]oxazolo[5,4-b]pyridin-6-one
3-(2-aminoethyl)-4-(5-chloro-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetic acid
4-(4-{[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(pyrazin-2-ylmethyl)-1,2-oxazole-3-carboxamide
1-(4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-phenylethan-1-ol
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(3-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]propanamide
3-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-N-(1-methyl-1H-imidazol-2-yl)benzamide
2-ethoxy-6-[({[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]phenol
1-[2-(dimethylamino)ethyl]-5-oxo-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrrolidine-3-carboxamide
2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
(2S)-2-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propanamide
(3-ethyl-1-phenylmethanesulfonylpiperidin-3-yl)methanol
{[2-(3,4-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}dimethylamine
1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
N-[2-(azepan-1-yl)ethyl]-N-(propan-2-yl)-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
9-(5-methylthiophene-3-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
methyl 2-chloro-4-{[(oxan-4-ylmethyl)carbamoyl]amino}benzoate
2-(3-ethylphenyl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
6-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-indole
(3S,4S)-1-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carbonyl]piperidine-3,4-diol
6-ethoxy-3-{[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1'-(2-hydroxypyridine-3-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-[({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]-6-methylpyridine-3-carbonitrile
4-{3-[5-(3-methylphenyl)-4-phenyl-1H-imidazol-1-yl]propyl}piperazin-2-one
5-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-cyclopentylpropanamide
3-{2-[(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)amino]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
{5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
N-[(2R,3R)-2-hydroxy-1'-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
(1S,6R)-3-methyl-4-oxo-N-(2,3,5-trifluorophenyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
(1S,4S)-2-(5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)-2-azabicyclo[2.2.1]heptane
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-3-ethoxypropan-1-one
(3aS,6aS)-2-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]piperazin-1-yl}ethan-1-ol
ethyl 4-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamido}piperidine-1-carboxylate
(2S,4R)-4-amino-1-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-(2-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
2-(5-{[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}furan-2-yl)benzonitrile
3-benzyl-4-[1-(propan-2-yl)-1H-pyrazole-3-carbonyl]piperazin-2-one
4-(4-chloro-3-methyl-1H-pyrazol-5-yl)-7-ethoxy-1,2,3,4-tetrahydroquinolin-2-one
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
N-cyclopropyl-2-{4-[(6-methoxypyrimidin-4-yl)amino]piperidin-1-yl}acetamide
2-(4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
(1R,3S)-7-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-ethoxy-7-azaspiro[3.5]nonan-1-ol
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethyl-1H-pyrrole-3-carboxamide